Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50009352
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  6.24E+8nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H L3A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  9.91E+8nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H K4A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527803(CHEMBL4557180)
Affinity DataEC50:  1.72E+5nMAssay Description:Binding affinity to human N-terminal His6-tagged human LDH-5 expressed in Escherichia coli Rosetta (DE3) assessed as induction of protein disruption ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527804(CHEMBL4453053)
Affinity DataKd:  1.78E+6nMAssay Description:Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) measured after 5 mins by Red-NHS fluor...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  1.01E+9nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H E5A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  9.54E+8nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H K6A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527805(CHEMBL4440124)
Affinity DataKd:  1.05E+6nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527806(CHEMBL4437918)
Affinity DataKd:  6.70E+4nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527807(CHEMBL4525659)
Affinity DataKd:  7.87E+5nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527808(CHEMBL4582140)
Affinity DataKd:  3.98E+5nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527809(CHEMBL4456178)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527810(CHEMBL4532326)
Affinity DataKd:  1.13E+5nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527811(CHEMBL4450669)
Affinity DataKd:  4.65E+5nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527803(CHEMBL4557180)
Affinity DataKd:  3.80E+5nMAssay Description:Competitive binding affinity to recombinant full length human His-tagged LDH-1 (1 to 322 residues) expressed in Escherichia coli assessed as protein-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527805(CHEMBL4440124)
Affinity DataKd:  1.02E+6nMAssay Description:Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) in sodium phosphate buffer at pH 7.6 b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527812(CHEMBL4475220)
Affinity DataKd:  1.49E+6nMAssay Description:Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) in sodium phosphate buffer at pH 7.6 b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  9.78E+8nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H T2A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527813(CHEMBL4456560)
Affinity DataKd:  6.40E+4nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527814(CHEMBL4471310)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527815(CHEMBL4468125)
Affinity DataKd:  1.42E+5nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527816(CHEMBL4452577)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527817(CHEMBL4466441)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  1.11E+9nMAssay Description:Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disruption by n...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataEC50:  2.33E+8nMAssay Description:Binding affinity full length human N-terminal His6-tagged LDH-H I8A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527803(CHEMBL4557180)
Affinity DataKd:  1.17E+5nMAssay Description:Competitive binding affinity to human N-terminal His6-tagged LDH-5 expressed in Escherichia coli Rosetta (DE3) assessed as protein-compound interacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527818(CHEMBL4575384)
Affinity DataKd:  1.05E+6nMAssay Description:Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) in sodium phosphate buffer at pH 7.6 b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50527803(CHEMBL4557180)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to truncated human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) after 5 mins by Red-NHS fluorescence dye...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed