Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50013735
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50397078(CHEMBL2171452)
Affinity DataKi:  3.70E+3nMAssay Description:Mixed type inhibition of human DNMT3A using AdoMet as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50397078(CHEMBL2171452)
Affinity DataKi:  5.03E+3nMAssay Description:Binding affinity to human DNMT3A catalytic domain assessed as inhibition of enzyme-mediated DNA methylation using 3H-AdoMet as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50427452(CHEMBL2326941)
Affinity DataKi:  9.16E+3nMAssay Description:Uncompetitive inhibition of human DNMT3A using AdoMet as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50427452(CHEMBL2326941)
Affinity DataKi:  1.14E+4nMAssay Description:Uncompetitive inhibition of human DNMT3A using poly dl-dC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50397078(CHEMBL2171452)
Affinity DataKi:  1.26E+4nMAssay Description:Mixed type inhibition of human DNMT3A using poly dl-dC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50427452(CHEMBL2326941)
Affinity DataKi:  1.38E+4nMAssay Description:Binding affinity to human DNMT3A catalytic domain assessed as inhibition of enzyme-mediated DNA methylation using 3H-AdoMet as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50427452(CHEMBL2326941)
Affinity DataKi:  1.61E+4nMAssay Description:Binding affinity to human DNMT3A catalytic domain assessed as inhibition of enzyme-mediated DNA methylation using poly dl-dC as substrate incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50397078(CHEMBL2171452)
Affinity DataKi:  2.16E+4nMAssay Description:Binding affinity to human DNMT3A catalytic domain assessed as inhibition of enzyme-mediated DNA methylation using poly dl-dC as substrate incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed