Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50014961
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 170nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 570nMAssay Description:Inhibition of OATP1B3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581556(CHEMBL5085260)
Affinity DataIC50: 600nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581557(CHEMBL5070789)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of OATP1B3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581555(CHEMBL5085115)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of MRP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPhosphatidylcholine translocator ABCB4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of MDR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581555(CHEMBL5085115)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581554(CHEMBL5092698)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of OATP1B3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581558(CHEMBL5083511)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of MRP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 3(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of MRP3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 3(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of MRP3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581553(CHEMBL5070166)
Affinity DataIC50: 3.54E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581554(CHEMBL5092698)
Affinity DataIC50: 4.63E+4nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of MRP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581553(CHEMBL5070166)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of BSEP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP2B6 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP2B6 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP3A4 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581551(CHEMBL5072201)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP3A4 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581552(Bms-986278 | BMS-986278)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP3A4 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50581550(Bms-986020 | AP-3152 FREE ACID | BMS-986020)
Affinity DataIC50: 5.00E+4nMAssay Description:Induction of CYP2C9 in human hepatocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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