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Found 19 Enz. Inhib. hit(s) with all data for entry = 50018518
TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataIC50:  370nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609079(CHEMBL5267793)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609092(CHEMBL5284829)
Affinity DataIC50:  3.61E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609085(CHEMBL5285095)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609080(CHEMBL5269273)
Affinity DataIC50:  4.17E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609075(CHEMBL5274041)
Affinity DataIC50:  4.69E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609084(CHEMBL5279065)
Affinity DataIC50:  5.15E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609090(CHEMBL5287258)
Affinity DataIC50:  5.81E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609086(CHEMBL5280426)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609078(CHEMBL5283312)
Affinity DataIC50:  6.35E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609087(CHEMBL5266258)
Affinity DataIC50:  6.78E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609076(CHEMBL5275819)
Affinity DataIC50:  6.94E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609088(CHEMBL5274196)
Affinity DataIC50:  7.48E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609082(CHEMBL5290468)
Affinity DataIC50:  9.89E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609089(CHEMBL5286176)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609081(CHEMBL5272408)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609091(CHEMBL5290556)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609077(CHEMBL5280193)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBromodomain-containing protein 4(Homo sapiens (Human))TBA
LigandPNGBDBM50609083(CHEMBL5288185)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) using C-terminal biotinylated tetra-acetylated histone H4 peptide as substrate incubated for 2.5 hrs by alpha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed