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Found 30 Enz. Inhib. hit(s) with all data for entry = 50015808
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589709(CHEMBL5173504)
Affinity DataKi:  4.40nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589713(CHEMBL5194064)
Affinity DataKi:  4.80nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589707(CHEMBL5171607)
Affinity DataKi:  7.70nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589716(CHEMBL5173926)
Affinity DataKi:  7.90nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589713(CHEMBL5194064)
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589715(CHEMBL5198312)
Affinity DataKi:  8.10nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589708(CHEMBL5186452)
Affinity DataKi:  9.80nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589714(CHEMBL5203770)
Affinity DataKi:  9.90nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589704(CHEMBL5171303)
Affinity DataKi:  10nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589712(CHEMBL5196435)
Affinity DataKi:  12nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589715(CHEMBL5198312)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  14nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589717(CHEMBL5176294)
Affinity DataKi:  15nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589706(CHEMBL5172461)
Affinity DataKi:  17nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589717(CHEMBL5176294)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589705(CHEMBL5191856)
Affinity DataKi:  19nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589707(CHEMBL5171607)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589710(CHEMBL5195262)
Affinity DataKi:  22nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589706(CHEMBL5172461)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589709(CHEMBL5173504)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589705(CHEMBL5191856)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589711(CHEMBL5183643)
Affinity DataKi:  37nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma-1 receptor in Sprague-Dawley rat cerebral membrane incubated for 90 mins by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589704(CHEMBL5171303)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589708(CHEMBL5186452)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589716(CHEMBL5173926)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589711(CHEMBL5183643)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589712(CHEMBL5196435)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589714(CHEMBL5203770)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50589710(CHEMBL5195262)
Affinity DataKi:  371nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membrane incubated for 90 mins in presence of by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed