Compile Data Set for Download or QSAR
Report error Found 1162 Enz. Inhib. hit(s) with all data for entry = 10754
LigandChemical structure of BindingDB Monomer ID 97529BDBM97529(US8470820, 40 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.0800nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 97514BDBM97514(US8470820, 25 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.0900nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 564307BDBM564307(Roche-Dataset for PDE10A, Compound 621)
Affinity DataIC50: 0.0900nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239752BDBM239752(US9394311, 35 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.150nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239837BDBM239837(US9394311, 119 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.170nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 97527BDBM97527(US8470820, 38 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.180nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563882BDBM563882(Roche-Dataset for PDE10A, Compound 196)
Affinity DataIC50: 0.190nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563870BDBM563870(Roche-Dataset for PDE10A, Compound 184)
Affinity DataIC50: 0.220nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239785BDBM239785(US9394311, 68 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.220nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239812BDBM239812(US9394311, 95 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.230nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 564109BDBM564109(Roche-Dataset for PDE10A, Compound 423)
Affinity DataIC50: 0.240nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239755BDBM239755(US9394311, 38 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.280nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239826BDBM239826(US9394311, 109 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.290nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563697BDBM563697(Roche-Dataset for PDE10A, Compound 11)
Affinity DataIC50: 0.300nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120583BDBM120583(US8703768, 183 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.300nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563771BDBM563771(Roche-Dataset for PDE10A, Compound 85)
Affinity DataIC50: 0.310nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120672BDBM120672(US8703768, 273 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.310nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120698BDBM120698(US8703768, 299 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.320nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563986BDBM563986(Roche-Dataset for PDE10A, Compound 300)
Affinity DataIC50: 0.330nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239840BDBM239840(US9394311, 122 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.350nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563700BDBM563700(Roche-Dataset for PDE10A, Compound 14)
Affinity DataIC50: 0.350nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563851BDBM563851(Roche-Dataset for PDE10A, Compound 165)
Affinity DataIC50: 0.360nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239838BDBM239838(US9394311, 120 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.360nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563881BDBM563881(Roche-Dataset for PDE10A, Compound 195)
Affinity DataIC50: 0.360nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120670BDBM120670(US8703768, 271 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.360nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120673BDBM120673(US8703768, 274 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.380nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120674BDBM120674(US8703768, 275 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.380nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120727BDBM120727(US8703768, 328 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.390nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120700BDBM120700(US8703768, 301 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.400nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120581BDBM120581(US8703768, 181 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.410nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239799BDBM239799(US9394311, 82 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.430nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120490BDBM120490(US8703768, 90 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.440nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239793BDBM239793(US9394311, 76 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.440nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239822BDBM239822(US9394311, 105 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.440nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563801BDBM563801(Roche-Dataset for PDE10A, Compound 115)
Affinity DataIC50: 0.450nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239753BDBM239753(US9394311, 36 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.470nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120624BDBM120624(US8703768, 225 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.480nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120489BDBM120489(US8703768, 89 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.480nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 200541BDBM200541(US9227970, 33 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.480nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120609BDBM120609(US8703768, 210 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.480nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120614BDBM120614(US8703768, 215 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.490nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239815BDBM239815(US9394311, 98 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.5nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 125040BDBM125040(US8772510, 59 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.510nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239823BDBM239823(US9394311, 106 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.540nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 239769BDBM239769(US9394311, 52 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.550nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120720BDBM120720(US8703768, 321 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.590nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563806BDBM563806(Roche-Dataset for PDE10A, Compound 120)
Affinity DataIC50: 0.600nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 563952BDBM563952(Roche-Dataset for PDE10A, Compound 266)
Affinity DataIC50: 0.600nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 317196BDBM317196(US9617271, 54 | 3,8-Dimethyl-6-((1-methyl-3-(pyrro...)
Affinity DataIC50: 0.640nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 120680BDBM120680(US8703768, 281 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.640nMAssay Description:Human PDE10A IC50 values were determined by using purified enzyme (Biomol cat. # SE-534) in a scintillation proximity assay (SPA) in 96 well plates (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2022
Entry Details Article
PubMed
Displayed 1 to 50 (of 1162 total ) | Next | Last >>
Jump to: