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Found 20 Enz. Inhib. hit(s) with all data for entry = 50018786
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  93nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50612554(CHEMBL5287581)
Affinity DataIC50:  144nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612554(CHEMBL5287581)
Affinity DataIC50:  160nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))TBA
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  196nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  235nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612554(CHEMBL5287581)
Affinity DataIC50:  245nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50612553(CHEMBL5271493)
Affinity DataIC50:  258nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612553(CHEMBL5271493)
Affinity DataIC50:  281nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612555(CHEMBL5281824)
Affinity DataIC50:  344nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612555(CHEMBL5281824)
Affinity DataIC50:  349nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50612556(CHEMBL5291493)
Affinity DataIC50:  458nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50612555(CHEMBL5281824)
Affinity DataIC50:  475nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612553(CHEMBL5271493)
Affinity DataIC50:  517nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612554(CHEMBL5287581)
Affinity DataIC50:  526nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  750nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612553(CHEMBL5271493)
Affinity DataIC50:  834nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612556(CHEMBL5291493)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50612556(CHEMBL5291493)
Affinity DataIC50:  1.63E+3nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612555(CHEMBL5281824)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50612556(CHEMBL5291493)
Affinity DataIC50:  3.85E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed