Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50015857
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590137(CHEMBL5198078)
Affinity DataIC50: 5.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590138(CHEMBL5201730)
Affinity DataIC50: 6.00E+3nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590137(CHEMBL5198078)
Affinity DataKd:  1.02E+4nMAssay Description:Binding affinity to CK2alpha (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590134(CHEMBL5180335)
Affinity DataIC50: 1.10E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590138(CHEMBL5201730)
Affinity DataKd:  1.58E+4nMAssay Description:Binding affinity to CK2alpha (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590135(CHEMBL5180822)
Affinity DataIC50: 1.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590136(CHEMBL5203610)
Affinity DataIC50: 1.90E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590133(CHEMBL5184713)
Affinity DataIC50: 8.60E+4nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50590132(CHEMBL5202453)
Affinity DataIC50: 3.33E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50099398(CHEMBL16425 | cid_761929 | 5-Bromo-1H-indazole)
Affinity DataIC50: 4.10E+5nMAssay Description:Negative allosteric modulation activity at CK2alpha (unknown origin) assessed as inhibition of CK2alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed