Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50018160
TargetMuscleblind-like protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405589BDBM50405589(CHEMBL1710607)
Affinity DataKd:  0.0110nMAssay Description:Binding affinity to MBNL1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMuscleblind-like protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 15236BDBM15236(CHEMBL164 | Cannabiscetin | 3,5,7-trihydroxy-2-(3,...)
Affinity DataKd:  0.25nMAssay Description:Binding affinity to MBNL1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234890BDBM50234890(CHEMBL4077018)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50550657BDBM50550657(CHEMBL4792737)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571459BDBM50571459(CHEMBL4872830)
Affinity DataKi:  1nMAssay Description:Binding affinity to ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059640BDBM50059640(CHEMBL2140173)
Affinity DataKi:  2nMAssay Description:Binding affinity to ATM (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039197BDBM50039197(1-Phenyl-cyclohexanecarboxylic acid 2-morpholin-4-...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to SIGMAR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMuscleblind-like protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405591BDBM50405591(CHEMBL5286270)
Affinity DataKd:  4nMAssay Description:Binding affinity to MBNL1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405622BDBM50405622(CHEMBL5271950)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405611BDBM50405611(CHEMBL5273419)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405622BDBM50405622(CHEMBL5271950)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHuntingtin(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595435BDBM50595435(CHEMBL5179682)
Affinity DataIC50: 8nMAssay Description:Inhibition of HTT (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20926BDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of HSP90alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50420459BDBM50420459(CHEMBL2086528)
Affinity DataIC50: 10nMAssay Description:Inhibition of TG2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50253320BDBM50253320(2-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-ylamin...)
Affinity DataIC50: 11nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50550657BDBM50550657(CHEMBL4792737)
Affinity DataKi:  15nMAssay Description:Binding affinity to Vps34 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405610BDBM50405610(CHEMBL5283014)
Affinity DataIC50: 17nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50059640BDBM50059640(CHEMBL2140173)
Affinity DataKi:  17nMAssay Description:Binding affinity to Vps34 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234888BDBM50234888(CHEMBL4074524)
Affinity DataIC50: 17nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405607BDBM50405607(CHEMBL5267784)
Affinity DataIC50: 17nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405605BDBM50405605(CHEMBL5273125)
Affinity DataIC50: 17nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405609BDBM50405609(CHEMBL5288429)
Affinity DataIC50: 17nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405608BDBM50405608(CHEMBL5274332)
Affinity DataIC50: 17nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103104BDBM50103104(CHEMBL3394106)
Affinity DataIC50: 18nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetKynurenine 3-monooxygenase(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50072083BDBM50072083(CHEMBL3407929)
Affinity DataIC50: 20nMAssay Description:Inhibition of KMO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHeat shock protein HSP 90-beta(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20926BDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50: 21nMAssay Description:Inhibition of HSP90beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405626BDBM50405626(CHEMBL5269500)
Affinity DataIC50: 24nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006932BDBM50006932(CHEMBL3237245)
Affinity DataIC50: 24nMAssay Description:Inhibition of KEAP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234888BDBM50234888(CHEMBL4074524)
Affinity DataIC50: 24nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405623BDBM50405623(CHEMBL5287474)
Affinity DataIC50: 26nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405624BDBM50405624(CHEMBL5284967)
Affinity DataIC50: 26nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405625BDBM50405625(CHEMBL5274433)
Affinity DataIC50: 29nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50103104BDBM50103104(CHEMBL3394106)
Affinity DataIC50: 30nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405623BDBM50405623(CHEMBL5287474)
Affinity DataIC50: 34nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234890BDBM50234890(CHEMBL4077018)
Affinity DataIC50: 36nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetKynurenine 3-monooxygenase(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061916BDBM50061916(3,4-Dimethoxy-N-[4-(3-nitro-phenyl)-thiazol-2-yl]-...)
Affinity DataIC50: 37nMAssay Description:Inhibition of KMO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHuntingtin(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595433BDBM50595433(CHEMBL5195936)
Affinity DataIC50: 40nMAssay Description:Inhibition of HTT (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405618BDBM50405618(CHEMBL5286810)
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetBDNF/NT-3 growth factors receptor(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405620BDBM50405620(CHEMBL5271538)
Affinity DataIC50: 47nMAssay Description:Inhibition of TrkB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405624BDBM50405624(CHEMBL5284967)
Affinity DataIC50: 48nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571459BDBM50571459(CHEMBL4872830)
Affinity DataKi:  50nMAssay Description:Binding affinity to Vps34 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50045333BDBM50045333(CHEBI:90705 | SB-203580)
Affinity DataIC50: 50nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHistone deacetylase 4(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405617BDBM50405617(CHEMBL5269131)
Affinity DataIC50: 54nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405621BDBM50405621(CHEMBL5283861)
Affinity DataIC50: 62nMAssay Description:Inhibition of TG2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405625BDBM50405625(CHEMBL5274433)
Affinity DataIC50: 74nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetHuntingtin(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595434BDBM50595434(CHEMBL5175104)
Affinity DataIC50: 80nMAssay Description:Inhibition of HTT (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMuscleblind-like protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405590BDBM50405590(CHEMBL5276958)
Affinity DataKd:  93nMAssay Description:Binding affinity to MBNL1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase 10(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405627BDBM50405627(CHEMBL5281537)
Affinity DataIC50: 94nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50405619BDBM50405619(CHEMBL5275178)
Affinity DataIC50: 98nMAssay Description:Inhibition of KEAP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Aligarh Muslim University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085415BDBM50085415(G6416 (GW5074) | 3-(3,5-dibromo-4-hydroxybenzylide...)
Affinity DataKd:  100nMAssay Description:Binding affinity to LC3B (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
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