Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50020646
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632292(CHEMBL5399029)
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632288(CHEMBL5432943 | US20250084074, Example 63)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632289(CHEMBL5410651)
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632291(CHEMBL5402640)
Affinity DataIC50: 19nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632275(CHEMBL5424226 | US20250084074, Example 38)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632295(CHEMBL5413808)
Affinity DataIC50: 39nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632288(CHEMBL5432943 | US20250084074, Example 63)
Affinity DataIC50: 51nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632286(CHEMBL5437239 | US20250084074, Example 143)
Affinity DataIC50: 61nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632270(CHEMBL5408867 | US20250084074, Example 4)
Affinity DataIC50: 63nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632291(CHEMBL5402640)
Affinity DataIC50: 66nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632275(CHEMBL5424226 | US20250084074, Example 38)
Affinity DataIC50: 86nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632279(CHEMBL5402097 | US20250084074, Example 219)
Affinity DataIC50: 89nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632292(CHEMBL5399029)
Affinity DataIC50: 90nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632282(CHEMBL5401191 | US20250084074, Example 133)
Affinity DataIC50: 93nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632274(CHEMBL5397143 | US20250084074, Example 34)
Affinity DataIC50: 101nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632294(CHEMBL5414939)
Affinity DataIC50: 107nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632270(CHEMBL5408867 | US20250084074, Example 4)
Affinity DataIC50: 109nMAssay Description:Displacement of FP-Probe from N-terminal His-tagged full length recombinant human HSET incubated for 2 hrs by fluorescence polarization based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632284(CHEMBL5398604 | US20250084074, Example 120)
Affinity DataIC50: 157nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50037967(CHEMBL3358270)
Affinity DataIC50: 171nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632293(CHEMBL5413274)
Affinity DataIC50: 217nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632259(CHEMBL5395577)
Affinity DataIC50: 257nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632273(CHEMBL5431102 | US20250084074, Example 37)
Affinity DataIC50: 260nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632290(CHEMBL5417430)
Affinity DataIC50: 260nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632287(CHEMBL5405412 | US20250084074, Example 142)
Affinity DataIC50: 288nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632259(CHEMBL5395577)
Affinity DataKd:  315nMAssay Description:Binding affinity to N-terminal His-tagged full length recombinant human HSET assessed as dissociation constant incubated for 3 hrs in presence of 7 u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632259(CHEMBL5395577)
Affinity DataKd:  332nMAssay Description:Binding affinity to N-terminal His-tagged full length recombinant human HSET assessed as dissociation constant incubated for 3 hrs in presence of 70 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632282(CHEMBL5401191 | US20250084074, Example 133)
Affinity DataIC50: 332nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632259(CHEMBL5395577)
Affinity DataKd:  371nMAssay Description:Binding affinity to N-terminal His-tagged full length recombinant human HSET assessed as dissociation constant by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataKd:  400nMAssay Description:Displacement of FP-Probe from N-terminal His-tagged full length recombinant human HSET incubated for 2 hrs by fluorescence polarization based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632281(CHEMBL5423487 | US20250084074, Example 141)
Affinity DataIC50: 405nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataKd:  436nMAssay Description:Displacement of FP-Probe from N-terminal His-tagged full length recombinant human HSET incubated for 2 hrs by fluorescence polarization based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50037967(CHEMBL3358270)
Affinity DataIC50: 825nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632271(CHEMBL5402598 | US20250084074, Example 36)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632262(CHEMBL5425236)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632269(CHEMBL5413665)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632260(CHEMBL5398248 | US20250084074, Example 1)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632268(CHEMBL5413268)
Affinity DataIC50: 3.54E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632261(CHEMBL5440441)
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632283(CHEMBL5435543)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50037967(CHEMBL3358270)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632280(CHEMBL5407106)
Affinity DataIC50: 4.44E+4nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632272(CHEMBL5435210)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632260(CHEMBL5398248 | US20250084074, Example 1)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632270(CHEMBL5408867 | US20250084074, Example 4)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632276(CHEMBL5425131)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632288(CHEMBL5432943 | US20250084074, Example 63)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIFC1(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632277(CHEMBL5414557)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of N-terminal His-tagged full length recombinant human HSET assessed as inhibition of microtubule-stimulated ATPase activity incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632291(CHEMBL5402640)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632275(CHEMBL5424226 | US20250084074, Example 38)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetKinesin-like protein KIF11(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50632282(CHEMBL5401191 | US20250084074, Example 133)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GST-tagged Eg5 (unknown origin) assessed as inhibition of microtubule-stimulated ATPase activity incubated for 80 mins in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
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