Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50020649
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: <1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 6nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 62nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: <100nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 134nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 148nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at human CAR LBD in human HepG2 cells incubated for 24 hrs by firefly luciferase reporter assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 3(Human)
Czech Academy of Sciences
Curated by ChEMBL
Czech Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 313nMAssay Description:Agonist activity at human recombinant GST-tagged CAR LBD incubated for 1 to 4 hrs in presence of fluorescein-labeled PGC1alpha by lanthascreen TR-FRE...More data for this Ligand-Target Pair








































