Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50018422
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM185171(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataKi:  150nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608169(CHEMBL5290129)
Affinity DataKi:  1.95E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608171(CHEMBL5268027)
Affinity DataKi:  2.32E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataKi:  3.98E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608174(CHEMBL5291124)
Affinity DataKi:  8.83E+3nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608175(CHEMBL5269953)
Affinity DataKi:  2.63E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608170(CHEMBL5278364)
Affinity DataKi:  3.06E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608167(CHEMBL5276215)
Affinity DataKi:  3.84E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608168(CHEMBL5266611)
Affinity DataKi:  6.18E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608172(CHEMBL5269861)
Affinity DataKi:  7.01E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608173(CHEMBL5282572)
Affinity DataKi:  8.85E+4nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50608176(CHEMBL5270888)
Affinity DataKi:  1.54E+5nMAssay Description:Reversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
University of Ottawa

Curated by ChEMBL
LigandPNGBDBM50073654(CHEBI:47807 | 4-(Methylsulfinyl)Butyl Isothiocyana...)
Affinity DataKi:  3.66E+5nMAssay Description:Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed