Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50022369
TargetTyrosinase(Human)TBA
LigandPNGBDBM50559076(CHEMBL4743159)
Affinity DataKi:  250nMAssay Description:Competitive inhibition of His-tagged human tyrosinase expressed in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50625100(CHEMBL5408197)
Affinity DataKi:  250nMAssay Description:Inhibition of human tyrosinaseMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataKi:  350nMAssay Description:Inhibition of human tyrosinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50559076(CHEMBL4743159)
Affinity DataKi:  920nMAssay Description:Binding affinity to human tyrosinase using l-DOPA as substrate assessed as inhibition constant by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50651532(CHEMBL5632644)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity to human tyrosinase using l-DOPA as substrate assessed as inhibition constant by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50559076(CHEMBL4743159)
Affinity DataIC50: 1.10E+3nMAssay Description:Competitive inhibition of His-tagged human tyrosinase expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50625100(CHEMBL5408197)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of tyrosinase in human MNT-1 cellsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPolyphenol oxidase 4(Agaricus bisporus)TBA
LigandPNGBDBM50651532(CHEMBL5632644)
Affinity DataIC50: 3.52E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50559076(CHEMBL4743159)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human tyrosinase using L-DOPA as substrate by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPolyphenol oxidase 4(Agaricus bisporus)TBA
LigandPNGBDBM50619201(CHEMBL4750140)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50651532(CHEMBL5632644)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human tyrosinase using L-DOPA as substrate by spectrophotometer analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50205807(CHEMBL3978212)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of tyrosinase in human MNT-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPolyphenol oxidase 4(Agaricus bisporus)TBA
LigandPNGBDBM50559076(CHEMBL4743159)
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetTyrosinase(Human)TBA
LigandPNGBDBM50619201(CHEMBL4750140)
Affinity DataIC50: 1.10E+6nMAssay Description:Inhibition of human tyrosinase using L-DOPA as substrate by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed