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TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50496545(CHEMBL3126804)
Affinity DataKi:  2nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652163(CHEMBL5642463)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human CA9 assessed as inhibition constant by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50496533(CHEMBL3126821)
Affinity DataKi:  2.80nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50130738(CHEMBL3633548)
Affinity DataKi:  6.5nMAssay Description:Binding affinity to human CA12 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652164(CHEMBL5639430)
Affinity DataKi:  7.80nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652164(CHEMBL5639430)
Affinity DataKi:  7.80nMAssay Description:Binding affinity to human CA12 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50130738(CHEMBL3633548)
Affinity DataKi:  14nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50588968(CHEMBL5189246)
Affinity DataKi:  19nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652167(CHEMBL5641923)
Affinity DataKi:  21nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50496534(CHEMBL3126817)
Affinity DataKi:  23nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50588968(CHEMBL5189246)
Affinity DataKi:  33nMAssay Description:Binding affinity to human CA12 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 37nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652149(CHEMBL5639934)
Affinity DataIC50: 38nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50496534(CHEMBL3126817)
Affinity DataKi:  44nMAssay Description:Binding affinity to human CA12 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652137(CHEMBL5646796)
Affinity DataIC50: 62nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652155(CHEMBL5647582)
Affinity DataIC50: 69nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652158(CHEMBL5646664)
Affinity DataIC50: 74nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652157(CHEMBL5647661)
Affinity DataIC50: 79nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652139(CHEMBL5639858)
Affinity DataIC50: 84nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652152(CHEMBL5646406)
Affinity DataIC50: 91nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652142(CHEMBL5639440)
Affinity DataIC50: 99nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652145(CHEMBL5646420)
Affinity DataIC50: 101nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652137(CHEMBL5646796)
Affinity DataIC50: 102nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652149(CHEMBL5639934)
Affinity DataIC50: 102nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652140(CHEMBL5646418)
Affinity DataIC50: 117nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652155(CHEMBL5647582)
Affinity DataIC50: 121nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652132(CHEMBL5646871)
Affinity DataIC50: 124nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652132(CHEMBL5646871)
Affinity DataIC50: 144nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652139(CHEMBL5639858)
Affinity DataIC50: 148nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652142(CHEMBL5639440)
Affinity DataIC50: 155nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652151(CHEMBL5646881)
Affinity DataIC50: 165nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652166(CHEMBL488481)
Affinity DataKi:  176nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652140(CHEMBL5646418)
Affinity DataIC50: 177nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652152(CHEMBL5646406)
Affinity DataIC50: 193nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652138(CHEMBL5639162)
Affinity DataIC50: 207nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652165(CHEMBL5647623)
Affinity DataKi:  225nMAssay Description:Binding affinity to human CA9 assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652158(CHEMBL5646664)
Affinity DataIC50: 240nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652145(CHEMBL5646420)
Affinity DataIC50: 246nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652136(CHEMBL5641726)
Affinity DataIC50: 247nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652150(CHEMBL5639472)
Affinity DataIC50: 276nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652138(CHEMBL5639162)
Affinity DataIC50: 317nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652157(CHEMBL5647661)
Affinity DataIC50: 354nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652151(CHEMBL5646881)
Affinity DataIC50: 354nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652136(CHEMBL5641726)
Affinity DataIC50: 363nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652156(CHEMBL5641721)
Affinity DataIC50: 367nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652146(CHEMBL5639588)
Affinity DataIC50: 379nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 12(Human)TBA
LigandPNGBDBM50652160(CHEMBL5647621)
Affinity DataIC50: 385nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652141(CHEMBL5647016)
Affinity DataIC50: 489nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCarbonic anhydrase 9(Human)TBA
LigandPNGBDBM50652150(CHEMBL5639472)
Affinity DataIC50: 492nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins followed by substrate addition and measured after 30 mins by spectrophotometric met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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