Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50021525
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]-epibatidine from human alpha3beta4 nAChRMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of [3H]-epibatidine from dopamine transporter (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [3H]-epibatidine from alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of [3H]-epibatidine from alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Displacement of [3H]-epibatidine from dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Noncompetitive inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:Displacement of [3H]-epibatidine from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Displacement of [3H]-epibatidine from alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Displacement of [3H]-epibatidine from sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-epibatidine from dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [3H]-epibatidine from alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]-epibatidine from human alpha2beta4 nAChRMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-epibatidine from alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]-epibatidine from dopamine transporter (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.46E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]-epibatidine from M2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]-epibatidine from M4 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of epibatidine-induced receptor activation at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as reduction in calcium flux preinc...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [3H]-epibatidine from M4 receptor (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 1.91E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois Chicago
Curated by ChEMBL
University of Illinois Chicago
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of nicotine induced calcium flux preincubated for 10 ...More data for this Ligand-Target Pair















