Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50020093 Sort by
LigandPNGBDBM50377863(AG-525 | CHEMBL257156)
Affinity DataKi:  277nMAssay Description:Displacement of [125I]apamin from SK2 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50241654((+)-berbamine | Berbamine | CHEMBL504323)
Affinity DataKi:  284nMAssay Description:Displacement of [125I]apamin from human SK2 expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50478473(CHEBI:49 | NSC-77037 | FANCHININ | Tetrandrine)
Affinity DataKi:  306nMAssay Description:Displacement of [125I]apamin from SK2 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50377863(AG-525 | CHEMBL257156)
Affinity DataKi:  370nMAssay Description:Displacement of [125I]apamin from SK3 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50478473(CHEBI:49 | NSC-77037 | FANCHININ | Tetrandrine)
Affinity DataKi:  461nMAssay Description:Displacement of [125I]apamin from SK3 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50241654((+)-berbamine | Berbamine | CHEMBL504323)
Affinity DataKi:  679nMAssay Description:Displacement of [125I]apamin from human SK3 expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50423643(CEPHARANTHINE)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [125I]apamin from human SK3 expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50626104(CHEMBL1182643)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]apamin from SK2 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50423643(CEPHARANTHINE)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [125I]apamin from human SK2 expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50626104(CHEMBL1182643)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [125I]apamin from SK3 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50626105(CHEMBL1185254)
Affinity DataKi:  1.69E+3nMAssay Description:Displacement of [125I]apamin from SK2 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50626105(CHEMBL1185254)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [125I]apamin from SK3 (unknown origin) expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed