Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50020599
LigandPNGBDBM50631733(CHEMBL5399711)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631732(CHEMBL5427972)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631731(CHEMBL5402284)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of VEGFR-2 (unknown origin) incubated for 45 mins by Kinase-Glo Max assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50631728(CHEMBL5409221)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of VEGFR-2 (unknown origin) incubated for 45 mins by Kinase-Glo Max assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50591689(CHEMBL5170911)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631753(CHEMBL5434391)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631755(CHEMBL5434570)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50591691(CHEMBL5175388)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50591690(CHEMBL5202279)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Srmpp

Curated by ChEMBL
LigandPNGBDBM50631763(CHEMBL5404166)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly Tyrosine peptide as substrate in presence of ATP incubated for 90 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631721(CHEMBL5418423)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant VEGFR-2 in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631739(CHEMBL5434432)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human recombinant VEGFR-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631740(CHEMBL5434411)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human recombinant VEGFR-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631754(CHEMBL5426655)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631722(CHEMBL5399297)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant VEGFR-2 in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631751(CHEMBL5396154)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant VEGFR-2 expressed in Sf21 insect cells incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50570077(CHEMBL4874971)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant VEGFR-2 in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631756(CHEMBL5397322)
Affinity DataIC50: 30nMAssay Description:Inhibition of human VEGFR-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50570076(CHEMBL4864168)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant VEGFR-2 in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631723(CHEMBL5422526)
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant VEGFR-2 in the presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631748(CHEMBL5410978)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631750(CHEMBL5438045)
Affinity DataIC50: 78nMAssay Description:Inhibition of human recombinant VEGFR-2 expressed in Sf21 insect cells incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631744(CHEMBL5407236)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Srmpp

Curated by ChEMBL
LigandPNGBDBM50631762(CHEMBL5427744)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly Tyrosine peptide as substrate in presence of ATP incubated for 90 mins by Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631745(CHEMBL5419219)
Affinity DataIC50: 83nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631749(CHEMBL5419779)
Affinity DataIC50: 86nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631746(CHEMBL5438926)
Affinity DataIC50: 95nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631747(CHEMBL5427270)
Affinity DataIC50: 102nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631736(CHEMBL5400653)
Affinity DataIC50: 199nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 60 mins by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631757(CHEMBL5433642)
Affinity DataIC50: 210nMAssay Description:Inhibition of human VEGFR-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631765(CHEMBL5395396)
Affinity DataIC50: 220nMAssay Description:Inhibition of VEGFR-2 (978 to 1408 residues) (unknown origin) using pEY (4:1) as substrate for 20 min in the presence of ATP by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631743(CHEMBL5421769)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Srmpp

Curated by ChEMBL
LigandPNGBDBM50631760(CHEMBL5408391)
Affinity DataIC50: 230nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631725(CHEMBL5430859)
Affinity DataIC50: 240nMAssay Description:Inhibition of VEGFR-2 (unknown origin) incubated for 45 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631742(CHEMBL5395478)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631741(CHEMBL5421530)
Affinity DataIC50: 280nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 346nMAssay Description:Inhibition of recombinant PDGFR-beta (unknown origin) incubated for 60 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetHepatocyte growth factor receptor(Human)
Srmpp

Curated by ChEMBL
LigandPNGBDBM50631761(CHEMBL5433522)
Affinity DataIC50: 360nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631735(CHEMBL5396774)
Affinity DataIC50: 386nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 60 mins by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631752(CHEMBL5402951)
Affinity DataIC50: 435nMAssay Description:Inhibition of recombinant PDGFR-beta (unknown origin) incubated for 60 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631724(CHEMBL5403714)
Affinity DataIC50: 480nMAssay Description:Inhibition of VEGFR-2 (unknown origin) incubated for 45 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631738(CHEMBL5420884)
Affinity DataIC50: 570nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 2.5 hrs by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631737(CHEMBL5435452)
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant VEGFR-2 kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate incubated for 2.5 hrs by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631766(CHEMBL5428581)
Affinity DataIC50: 820nMAssay Description:Inhibition of VEGFR-2 (978 to 1408 residues) (unknown origin) using pEY (4:1) as substrate for 20 min in the presence of ATP by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631764(CHEMBL5423804)
Affinity DataIC50: 910nMAssay Description:Inhibition of VEGFR-2 (978 to 1408 residues) (unknown origin) using pEY (4:1) as substrate for 20 min in the presence of ATP by ELISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631729(CHEMBL5427272)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 5 mins by ELISA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM50631730(CHEMBL5404662)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 5 mins by ELISA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of VEGFR-2 (unknown origin) kinase activity using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 5 mins by ELISA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Srmpp

Curated by ChEMBL
LigandPNGBDBM50510881(CHEMBL4515066)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of c-Met (unknown origin) using poly(Glu-Tyr) at 4:1 ratio as substrate in presence of ATP incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
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