Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50021944
Affinity DataKd: 28nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 49nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 55nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 56nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 127nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 145nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 183nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataKd: 666nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 679nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 777nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataKd: 841nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.16E+3nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 4.09E+3nMAssay Description:Binding affinity to human DNMT1 in presence of 10 uM SAM by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.15E+3nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataIC50: 3.82E+4nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of DNMT1 (unknown origin) using semi-methylated DNA substrate preincubated for 15 mins followed by substrate and [3H-SAM] addition and mea...More data for this Ligand-Target Pair
Affinity DataKd: 9.46E+4nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli assessed as equilibrium dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 9.46E+4nMAssay Description:Binding affinity to human DNMT1 expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair









