Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50021868
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  1nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  1nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  2nMAssay Description:Binding affinity to BRDT BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  2.80nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  3nMAssay Description:Binding affinity to BRDT BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  7.40nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645659(CHEMBL5590267)
Affinity DataIC50: 11nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataIC50: 12nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  14nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataIC50: 15nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 17nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645660(CHEMBL5591911)
Affinity DataIC50: 18nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645659(CHEMBL5590267)
Affinity DataIC50: 20nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  26nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645657(CHEMBL5583993)
Affinity DataIC50: 27nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  29nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50560174(GSK789)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645662(CHEMBL5594256)
Affinity DataIC50: 53nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645655(CHEMBL5596020)
Affinity DataIC50: 63nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50560174(GSK789)
Affinity DataIC50: 77nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 85nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  86nMAssay Description:Binding affinity to BRDT BD1 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645663(CHEMBL5590506)
Affinity DataIC50: 150nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645664(CHEMBL5593005)
Affinity DataIC50: 180nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataIC50: 180nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  250nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataIC50: 260nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  260nMAssay Description:Binding affinity to BRD3 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  510nMAssay Description:Binding affinity to BRD2 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  530nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645655(CHEMBL5596020)
Affinity DataIC50: 650nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  660nMAssay Description:Binding affinity to BRD3 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645658(CHEMBL5590067)
Affinity DataKd:  680nMAssay Description:Binding affinity to BRDT BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  770nMAssay Description:Binding affinity to BRD2 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataIC50: 770nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645657(CHEMBL5583993)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645660(CHEMBL5591911)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645656(CHEMBL5590913)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to BRDT BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645664(CHEMBL5593005)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  6.50E+3nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645663(CHEMBL5590506)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  9.80E+3nMAssay Description:Binding affinity to BRD3 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to BRDT BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645661(CHEMBL5590578)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRD2 BD2 (unknown origin) assessed as dissociation constant by BROMOscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50645662(CHEMBL5594256)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50560174(GSK789)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50560174(GSK789)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed