Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50021375
TargetHeparanase(Human)TBA
LigandPNGBDBM50640013(CHEMBL5562364)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640011(CHEMBL5559476)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640010(CHEMBL5561988)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640009(CHEMBL5549928)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640004(CHEMBL5557429)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640007(CHEMBL5556661)
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640012(CHEMBL5557768)
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640006(CHEMBL5559840)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640003(CHEMBL5564261)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640005(CHEMBL5560024)
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640008(CHEMBL5559647)
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640002(CHEMBL5561039)
Affinity DataIC50: 92nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50388331(CHEMBL2059499)
Affinity DataIC50: 123nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSpike glycoprotein(2019-nCoV)TBA
LigandPNGBDBM50640006(CHEMBL5559840)
Affinity DataKd:  1.87E+3nMAssay Description:Binding affinity to RBD domain of SARS-CoV-2 spike protein assessed as dissociation constant by Isothermal Titration CalorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSpike glycoprotein(2019-nCoV)TBA
LigandPNGBDBM50640000(CHEMBL5568325)
Affinity DataKd:  2.11E+3nMAssay Description:Binding affinity to RBD domain of SARS-CoV-2 spike protein assessed as dissociation constant by Isothermal Titration CalorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640001(CHEMBL5567072)
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50639998(CHEMBL5560742)
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50640000(CHEMBL5568325)
Affinity DataIC50: 3.44E+3nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50639997(CHEMBL5561651)
Affinity DataIC50: 3.54E+3nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSpike glycoprotein(2019-nCoV)TBA
LigandPNGBDBM50388331(CHEMBL2059499)
Affinity DataKd:  9.12E+3nMAssay Description:Binding affinity to RBD domain of SARS-CoV-2 spike protein assessed as dissociation constant by Isothermal Titration CalorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSpike glycoprotein(2019-nCoV)TBA
LigandPNGBDBM50639997(CHEMBL5561651)
Affinity DataKd:  9.18E+3nMAssay Description:Binding affinity to RBD domain of SARS-CoV-2 spike protein assessed as dissociation constant by Isothermal Titration CalorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeparanase(Human)TBA
LigandPNGBDBM50639999(CHEMBL5568403)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of recombinant human heparanase expressed in Insect cells assessed as fondaparinux cleavage by measuring disaccharide product incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed