Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50022153
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in CHO cells cotransfected with genetic response element-luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648666(CHEMBL5611927)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648654(CHEMBL5612987)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in CHO cells cotransfected with genetic response element-luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648654(CHEMBL5612987)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648669(CHEMBL5614270)
Affinity DataIC50: 69nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648660(CHEMBL5614066)
Affinity DataIC50: 113nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 131nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648669(CHEMBL5614270)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648654(CHEMBL5612987)
Affinity DataIC50: 162nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648669(CHEMBL5614270)
Affinity DataIC50: 174nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648666(CHEMBL5611927)
Affinity DataIC50: 196nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648654(CHEMBL5612987)
Affinity DataIC50: 209nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648680(CHEMBL5612826)
Affinity DataIC50: 268nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648660(CHEMBL5614066)
Affinity DataIC50: 274nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648660(CHEMBL5614066)
Affinity DataIC50: 291nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648660(CHEMBL5614066)
Affinity DataIC50: 401nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648661(CHEMBL5611949)
Affinity DataIC50: 441nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648669(CHEMBL5614270)
Affinity DataIC50: 443nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648673(CHEMBL5612599)
Affinity DataIC50: 447nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648677(CHEMBL5614351)
Affinity DataIC50: 532nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648665(CHEMBL5614193)
Affinity DataIC50: 541nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648667(CHEMBL5612373)
Affinity DataIC50: 608nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648671(CHEMBL5611932)
Affinity DataIC50: 653nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648656(CHEMBL5613136)
Affinity DataIC50: 672nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648668(CHEMBL5612249)
Affinity DataIC50: 697nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648666(CHEMBL5611927)
Affinity DataIC50: 831nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648657(CHEMBL5612088)
Affinity DataIC50: 953nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648655(CHEMBL5612610)
Affinity DataIC50: 1.03E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648674(CHEMBL5613366)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648681(CHEMBL5613738)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648678(CHEMBL5613159)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648662(CHEMBL5613719)
Affinity DataIC50: 1.27E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648659(CHEMBL5612444)
Affinity DataIC50: 1.45E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648682(CHEMBL5613491)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648672(CHEMBL5613699)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648683(CHEMBL5612255)
Affinity DataIC50: 1.93E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648676(CHEMBL5612843)
Affinity DataIC50: 1.98E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648658(CHEMBL5613411)
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648663(CHEMBL5612482)
Affinity DataIC50: 2.98E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648675(CHEMBL5613281)
Affinity DataIC50: 3.09E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648664(CHEMBL5611909)
Affinity DataIC50: 3.68E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648679(CHEMBL5612979)
Affinity DataIC50: 3.86E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648666(CHEMBL5611927)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed