Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50022799
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654424BDBM50654424(CHEMBL6142132)
Affinity DataIC50: 10nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654427BDBM50654427(CHEMBL6103202)
Affinity DataIC50: 37nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654423BDBM50654423(CHEMBL6149594)
Affinity DataIC50: 75nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654428BDBM50654428(CHEMBL6120620)
Affinity DataIC50: 75nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654430BDBM50654430(CHEMBL6133368)
Affinity DataIC50: 75nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654425BDBM50654425(CHEMBL6143158)
Affinity DataIC50: 100nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654422BDBM50654422(CHEMBL6096615)
Affinity DataIC50: 100nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654429BDBM50654429(CHEMBL6147299)
Affinity DataIC50: 100nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetHeparanase(Human)
Istituto di Ricerche Chimiche e Biochimiche G. Ronzoni

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654426BDBM50654426(CHEMBL6142214)
Affinity DataIC50: 100nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed