Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50023043
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Binding affinity to QPTCL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of QPCT (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: <2nMAssay Description:Binding affinity to QPTCL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of QPCT (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to QPTCL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to QPTCL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: <25nMAssay Description:Binding affinity to QPTCL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of QPCT (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: <100nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of QPCT (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of QPCT (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 5.70E+3nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.10E+3nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 7.30E+3nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKd: 9.40E+3nMAssay Description:Binding affinity to QPCTL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataIC50: 5.09E+4nMAssay Description:Inhibition of QPCTL (unknown origin)More data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 7.90E+4nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 9.50E+4nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.03E+5nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+5nMAssay Description:Binding affinity to QPCT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 1.99E+5nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Tongji University Cancer Center
Curated by ChEMBL
Tongji University Cancer Center
Curated by ChEMBL
Affinity DataKi: 2.19E+5nMAssay Description:Binding affinity to QPCTL (unknown origin) extracted from Escherichia coli BL21 (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair














3D Structure (crystal)






