Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50023188
TargetSRSF protein kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660191BDBM50660191(CHEMBL6170692)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of SRPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660192BDBM50660192(CHEMBL6166766)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of 6His/SUMO- tagged human ABL1 (229 to 500 residues) extracted from Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProteasome subunit beta type-7(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660190BDBM50660190(CHEMBL6143686)
Affinity DataIC50: 3.40nMAssay Description:Activation of 26s proteosome (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50638111BDBM50638111(CHEMBL5517884)
Affinity DataIC50: 27nMAssay Description:Inhibition of MCL-1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSRSF protein kinase 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512854BDBM50512854(CHEMBL4468747 | US11066363, Compound 37)
Affinity DataIC50: 36nMAssay Description:Inhibition of SRPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660193BDBM50660193(CHEMBL6149601)
Affinity DataIC50: 48nMAssay Description:Inhibition of EGFR (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660188BDBM50660188(CHEMBL6146781)
Affinity DataIC50: 60nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCyclin-dependent kinase 3(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660187BDBM50660187(CHEMBL5086595)
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant CDK3 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSRSF protein kinase 2(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50512854BDBM50512854(CHEMBL4468747 | US11066363, Compound 37)
Affinity DataIC50: 98nMAssay Description:Inhibition of SRPK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCyclin-dependent kinase 12(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660187BDBM50660187(CHEMBL5086595)
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant CDK12 (unknown origin) extracted from baculovirus infected insect cellsMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCathepsin G(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660194BDBM50660194(CHEMBL6171603)
Affinity DataIC50: 190nMAssay Description:Inhibition of human Cathepsin GMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCathepsin G(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610524BDBM50610524(CHEMBL5274237)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Cathepsin GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 178123BDBM178123((2'R*,7R*)-3-(4-methoxybenzyl)-3,5,6,7-tetrahy...)
Affinity DataIC50: 220nMAssay Description:Inhibition of MetAP2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetNeutrophil elastase(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610524BDBM50610524(CHEMBL5274237)
Affinity DataIC50: 240nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetProtein cereblon(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50614095BDBM50614095(CHEMBL304572)
Affinity DataIC50: 605nMAssay Description:Inhibition of CRBN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660189BDBM50660189(CHEMBL6168711)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of c-KIT (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetNeutrophil elastase(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660194BDBM50660194(CHEMBL6171603)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCyclin-dependent kinase 7(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50110178BDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetCyclin-dependent kinase 7(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50660187BDBM50660187(CHEMBL5086595)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetGTPase KRas(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50623207BDBM50623207(CHEMBL5419780)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity to human KRAS G12S mutant assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed