Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029165
LigandPNGBDBM50281909((R)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  1.5nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281903((S)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  2.20nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281902((R)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  2.70nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281902((R)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281909((R)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  3.20nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281906(2-[(E)-2-(9,9a-Dihydro-4aH-xanthen-9-yl)-vinyl]-1-...)
Affinity DataKd:  3.40nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281903((S)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  4.90nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281903((S)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  4.92nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281905(2-[3-(10H-Anthracen-9-ylidene)-propyl]-1-methyl-pi...)
Affinity DataKd:  5nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281904(2-[(E)-3-(9,10-Dihydro-anthracen-9-yl)-allyl]-1-me...)
Affinity DataKd:  5.20nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281905(2-[3-(10H-Anthracen-9-ylidene)-propyl]-1-methyl-pi...)
Affinity DataKd:  7.60nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((1S,2R,6S)-1,6-D...)
Affinity DataKd:  9.10nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281902((R)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  12nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281902((R)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  15nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281903((S)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-...)
Affinity DataKd:  21nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281904(2-[(E)-3-(9,10-Dihydro-anthracen-9-yl)-allyl]-1-me...)
Affinity DataKd:  23nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281907((S)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  24nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281906(2-[(E)-2-(9,9a-Dihydro-4aH-xanthen-9-yl)-vinyl]-1-...)
Affinity DataKd:  25nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281907((S)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl...)
Affinity DataKd:  35nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((1S,2R,6S)-1,6-D...)
Affinity DataKd:  168nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281908(2-((E)-2-Anthracen-9-yl-vinyl)-1-methyl-piperidine...)
Affinity DataKd:  635nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281908(2-((E)-2-Anthracen-9-yl-vinyl)-1-methyl-piperidine...)
Affinity DataKd:  679nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50280521((4R,5S)-5-Methyl-4-[(E)-3-((R)-1-methyl-piperidin-...)
Affinity DataKd:  1.21E+3nMAssay Description:Displacement of [3H]QNB from rat brain stem muscarinic receptor 2 (M2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50280521((4R,5S)-5-Methyl-4-[(E)-3-((R)-1-methyl-piperidin-...)
Affinity DataKd:  9.70E+3nMAssay Description:Displacement of [3H]QNB from muscarinic receptor 1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article