Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50029286
LigandChemical structure of BindingDB Monomer ID 50031491BDBM50031491(3-(2'-Propylaminocarbonylsulfamoyl-biphenyl-4-ylme...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283002BDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283000BDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50032362BDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50032364BDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032362BDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283001BDBM50283001(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283005BDBM50283005(3-(2'-Butyloxycarbonylsulfamoyl-3-bromo-biphenyl-4...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 36645BDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283003BDBM50283003(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283000BDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283006BDBM50283006(3-(2'-Butyloxycarbonylsulfamoyl-biphenyl-4-ylmethy...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283008BDBM50283008(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50049179BDBM50049179(L-161570 | 4'-(4-Ethyl-5-formyl-2-propyl-imidazol-...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032364BDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 82428BDBM82428(CAS_124750-95-4 | CB91356279 | CHEMBL443269 | DuP ...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50032351BDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283009BDBM50283009(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50049196BDBM50049196(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283007BDBM50283007(3-(2'-Butyloxycarbonylsulfamoyl-3-methyl-biphenyl-...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283002BDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50282999BDBM50282999(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283004BDBM50283004(5-Ethyl-3-[3-fluoro-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283012BDBM50283012(3-(2'-Butyloxycarbonylsulfamoyl-3-nitro-biphenyl-4...)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032351BDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283009BDBM50283009(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283013BDBM50283013(3-[3-Chloro-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283007BDBM50283007(3-(2'-Butyloxycarbonylsulfamoyl-3-methyl-biphenyl-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283001BDBM50283001(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282999BDBM50282999(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283003BDBM50283003(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283012BDBM50283012(3-(2'-Butyloxycarbonylsulfamoyl-3-nitro-biphenyl-4...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283005BDBM50283005(3-(2'-Butyloxycarbonylsulfamoyl-3-bromo-biphenyl-4...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283010BDBM50283010(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283011BDBM50283011(5-Ethyl-3-[3-methyl-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283006BDBM50283006(3-(2'-Butyloxycarbonylsulfamoyl-biphenyl-4-ylmethy...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049196BDBM50049196(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 80nMAssay Description:Compound was tested for the inhibition of angiotensin II AT2 receptor by displacement of [125I]- Ang II to rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283008BDBM50283008(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50: 80nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049179BDBM50049179(L-161570 | 4'-(4-Ethyl-5-formyl-2-propyl-imidazol-...)
Affinity DataIC50: 500nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283013BDBM50283013(3-[3-Chloro-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 500nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283010BDBM50283010(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50: 700nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031491BDBM50031491(3-(2'-Propylaminocarbonylsulfamoyl-biphenyl-4-ylme...)
Affinity DataIC50: 775nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283011BDBM50283011(5-Ethyl-3-[3-methyl-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283004BDBM50283004(5-Ethyl-3-[3-fluoro-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82428BDBM82428(CAS_124750-95-4 | CB91356279 | CHEMBL443269 | DuP ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36645BDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article