Compile Data Set for Download or QSAR
maximum 50k data
Found 51 Enz. Inhib. hit(s) with all data for entry = 50029431
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284388(2-{[Acetyl-(1-hexadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataKi:  1.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284401(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284395(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataKi:  6.60nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataKi:  7.20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284399(1-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataKi:  9.40nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284409(2-{[Acetyl-(2,2-dimethyl-3-octadecylcarbamoyloxy-p...)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284386(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataKi:  20nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataKi:  23nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284398(3-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284392(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataKi:  30nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284396(3-[5-(3-Octadecylcarbamoyloxymethyl-oxetan-3-ylmet...)
Affinity DataKi:  31nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284387(3-[5-(3-Hexadecyloxymethyl-oxetan-3-ylmethoxycarbo...)
Affinity DataKi:  53nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284403(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclohex...)
Affinity DataKi:  56nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284394(2-{[Acetyl-(3-hexadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataKi:  95nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284407(2-{[Acetyl-(3-hexadecyloxymethyl-oxetan-3-ylmethox...)
Affinity DataKi:  110nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284402(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclohep...)
Affinity DataKi:  110nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284406(1-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataKi:  112nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284405(3-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataKi:  139nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284404(1-[5-(3-Octadecylcarbamoyloxymethyl-oxetan-3-ylmet...)
Affinity DataKi:  188nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284397(2-{[Acetyl-(1-acetyl-3-hexadecylcarbamoyloxymethyl...)
Affinity DataKi:  278nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284390(1-[5-(3-Hexadecyloxymethyl-thietan-3-ylmethoxycarb...)
Affinity DataKi:  596nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284393(CHEMBL11731 | Heterocyclic Lipid derivative)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284389(CHEMBL12055 | Heterocyclic Lipid derivative)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284391(1-[5-(3-Hexadecyloxymethyl-oxetan-3-ylmethoxycarbo...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-PAF from its Platelet Activating Factor (PAF) receptor in rabbit platelet membrane in vitro.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284392(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284394(2-{[Acetyl-(3-hexadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataIC50:  93nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284399(1-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataIC50:  95nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284395(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataIC50:  118nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataIC50:  123nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284400(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-oxetan-3...)
Affinity DataIC50:  158nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284397(2-{[Acetyl-(1-acetyl-3-hexadecylcarbamoyloxymethyl...)
Affinity DataIC50:  188nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284407(2-{[Acetyl-(3-hexadecyloxymethyl-oxetan-3-ylmethox...)
Affinity DataIC50:  219nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284386(1-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataIC50:  228nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284398(3-[5-(3-Octadecylcarbamoyloxymethyl-thietan-3-ylme...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284403(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclohex...)
Affinity DataIC50:  286nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284388(2-{[Acetyl-(1-hexadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284402(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclohep...)
Affinity DataIC50:  365nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284396(3-[5-(3-Octadecylcarbamoyloxymethyl-oxetan-3-ylmet...)
Affinity DataIC50:  382nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284409(2-{[Acetyl-(2,2-dimethyl-3-octadecylcarbamoyloxy-p...)
Affinity DataIC50:  394nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50251276(BN 52021 | CHEMBL514432 | GINKOLIDE B | Gingkolide...)
Affinity DataIC50:  418nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284401(2-{[Acetyl-(1-octadecylcarbamoyloxymethyl-cyclopen...)
Affinity DataIC50:  573nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284390(1-[5-(3-Hexadecyloxymethyl-thietan-3-ylmethoxycarb...)
Affinity DataIC50:  658nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284404(1-[5-(3-Octadecylcarbamoyloxymethyl-oxetan-3-ylmet...)
Affinity DataIC50:  684nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284405(3-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataIC50:  1.14E+3nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284387(3-[5-(3-Hexadecyloxymethyl-oxetan-3-ylmethoxycarbo...)
Affinity DataIC50:  1.26E+3nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284389(CHEMBL12055 | Heterocyclic Lipid derivative)
Affinity DataIC50:  1.27E+3nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284406(1-[4-(1-Octadecylcarbamoyloxymethyl-cyclopentylmet...)
Affinity DataIC50:  1.45E+3nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284391(1-[5-(3-Hexadecyloxymethyl-oxetan-3-ylmethoxycarbo...)
Affinity DataIC50:  1.47E+3nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails Article
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: