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Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50037775
TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50002694(MOTILIN)
Affinity DataKi:  0.360nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199368((9R,12R,15S)-12-isopropyl-9-(4-methoxy-benzyl)-15-...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199372((9R,12R,15S)-12-isopropyl-9-naphthalen-1-ylmethyl-...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199359((9R,12R,15S)-9-benzo[b]thiophen-3-ylmethyl-12-isop...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199397((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199347((9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8...)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199353((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-i...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199373((9R,12R,15S)-9-benzyl-12-isopropyl-15-propyl-6,7,8...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199396((9R,12R,15S)-12-isopropyl-9-naphthalen-2-ylmethyl-...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199365((E)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl...)
Affinity DataKi:  137nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199362((9R,12R,15S)-15-benzyl-9-(4-hydroxy-benzyl)-12-iso...)
Affinity DataKi:  185nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199394((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  192nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199364((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-methyl-15-pro...)
Affinity DataKi:  196nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199392((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-isobutyl-12-i...)
Affinity DataKi:  222nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199346((9R,12R,15S)-9-(1H-indol-3-ylmethyl)-12-isopropyl-...)
Affinity DataKi:  255nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199390((9R,12R,15R)-9-(4-Hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  335nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199376((9R,12R,15S)-9-(4-hydroxy-benzyl)-15-hydroxymethyl...)
Affinity DataKi:  650nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199378((9R,12R,15S)-15-(4-amino-butyl)-9-(4-hydroxy-benzy...)
Affinity DataKi:  664nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199349((E)-(3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-...)
Affinity DataKi:  701nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199361((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  982nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199360((3S,6R,9R)-9-(4-hydroxy-benzyl)-6-isopropyl-3-prop...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199351((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199363((9R,12R,15S)-12-isopropyl-9-phenethyl-15-propyl-6,...)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199377((9R,12R,15S)-12-benzyl-9-(4-hydroxy-benzyl)-15-pro...)
Affinity DataKi:  1.52E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199389((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  1.88E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199352((9R,13R,16S)-9-(4-hydroxy-benzyl)-13-isopropyl-16-...)
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199382((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-10,...)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199391((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-8-m...)
Affinity DataKi:  2.78E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199385((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199350((9R,12R,15S)-9-cyclohexylmethyl-12-isopropyl-15-pr...)
Affinity DataKi:  3.25E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199388((9R,12R,15S)-9,12-diisopropyl-15-propyl-6,7,8,9,11...)
Affinity DataKi:  3.57E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199383(3-[(9R,12R,15S)-9-(4-hydroxy-benzyl)-10,13,16-trio...)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199357((9S,12R,15R)-15-(4-hydroxy-benzyl)-12-isopropyl-9-...)
Affinity DataKi:  6.06E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199358((8R,11R,14S)-8-(4-hydroxy-benzyl)-11-isopropyl-14-...)
Affinity DataKi:  6.06E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199366((9R,12R,15S)-8-acetyl-9-(4-hydroxy-benzyl)-12-isop...)
Affinity DataKi:  6.39E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199374((E/Z)-(9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isoprop...)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199393((E/Z)-(8R,11R,14S)-8-(4-Hydroxy-benzyl)-11-isoprop...)
Affinity DataKi:  9.73E+3nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199386((9R,12R,15S)-9-(4-amino-butyl)-12-isopropyl-15-pro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199395((S)-2-((R)-2-((R)-2-(2-(2-((E)-3-acetamidoprop-1-e...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199387((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-11-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199384((9R,12R,15S)-12-isopropyl-9-methyl-15-propyl-6,7,8...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199381((9S,12R,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199375((10S,13R,16R)-16-(4-hydroxy-benzyl)-13-isopropyl-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199379((E/Z)-(8R,11R,14S)-8-(4-hydroxy-benzyl)-11-isoprop...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199380((9R,12R,15S)-12-isopropyl-9-phenyl-15-propyl-6,7,8...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199370((7R,10R,13S)-7-(4-hydroxy-benzyl)-10-isopropyl-13-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199369((9R,12S,15S)-9-(4-hydroxy-benzyl)-12-isopropyl-15-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199367((9R,12R,15S)-9-(4-hydroxy-benzyl)-12-hydroxymethyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199356((S)-2-((R)-2-((R)-2-amino-3-(4-hydroxyphenyl)propa...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMotilin receptor(Human)
Tranzyme Pharma

Curated by ChEMBL
LigandPNGBDBM50199354((9S,12R,15R)-15-(4-hydroxy-benzyl)-12-isopropyl-9-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]motilin from human MOTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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