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Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50036359
TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453787(CHEMBL2113556)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453793(CHEMBL2113559)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50368489(CHEMBL611571)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453790(CHEMBL2113563)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453789(CHEMBL2113564)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453788(CHEMBL2113558)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453792(CHEMBL2113560)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453796(CHEMBL2113552)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453791(CHEMBL2113555)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453795(CHEMBL2113553)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453795(CHEMBL2113553)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453794(CHEMBL2113554)
Affinity DataKi:  264nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453794(CHEMBL2113554)
Affinity DataKi:  384nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453792(CHEMBL2113560)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453787(CHEMBL2113556)
Affinity DataKi:  524nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453793(CHEMBL2113559)
Affinity DataKi:  545nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataKi:  569nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453788(CHEMBL2113558)
Affinity DataKi:  935nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453796(CHEMBL2113552)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453790(CHEMBL2113563)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453791(CHEMBL2113555)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50368489(CHEMBL611571)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453789(CHEMBL2113564)
Affinity DataKi:  1.85E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453787(CHEMBL2113556)
Affinity DataEC50: >10nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453788(CHEMBL2113558)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453790(CHEMBL2113563)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453789(CHEMBL2113564)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50368489(CHEMBL611571)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453790(CHEMBL2113563)
Affinity DataEC50:  269nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453789(CHEMBL2113564)
Affinity DataEC50:  195nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453793(CHEMBL2113559)
Affinity DataEC50:  4.89E+3nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453793(CHEMBL2113559)
Affinity DataEC50:  281nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453787(CHEMBL2113556)
Affinity DataEC50:  482nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453791(CHEMBL2113555)
Affinity DataEC50:  800nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453788(CHEMBL2113558)
Affinity DataEC50:  638nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453792(CHEMBL2113560)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50368489(CHEMBL611571)
Affinity DataEC50:  747nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453792(CHEMBL2113560)
Affinity DataEC50:  677nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataEC50:  8.20nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  55nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  394nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453791(CHEMBL2113555)
Affinity DataEC50:  4.34E+3nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50453794(CHEMBL2113554)
Affinity DataEC50:  1.97E+3nMAssay Description:Activitty at Adenosine A1 receptor of rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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