Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50006117
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140906BDBM50140906(1-[2-[1-[2-amino-3-(4-hydroxyphenyl)-(2S)-propanoy...)
Affinity DataIC50: 21nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456337BDBM50456337(CHEMBL267708)
Affinity DataIC50: 29nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456336BDBM50456336(CHEMBL2371360)
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456335BDBM50456335(CHEMBL2371359)
Affinity DataIC50: 109nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456332BDBM50456332(CHEMBL2371339)
Affinity DataIC50: 170nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456336BDBM50456336(CHEMBL2371360)
Affinity DataIC50: 202nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166066BDBM50166066(CHEMBL362991 | Tyr-Pro-Phe-Pro-NH2 | [D-Pro4]morph...)
Affinity DataIC50: 552nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456334BDBM50456334(CHEMBL2371340)
Affinity DataIC50: 557nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456335BDBM50456335(CHEMBL2371359)
Affinity DataIC50: 594nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140906BDBM50140906(1-[2-[1-[2-amino-3-(4-hydroxyphenyl)-(2S)-propanoy...)
Affinity DataIC50: 1.25E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456337BDBM50456337(CHEMBL267708)
Affinity DataIC50: 1.51E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456332BDBM50456332(CHEMBL2371339)
Affinity DataIC50: 1.79E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456339BDBM50456339(CHEMBL2371336)
Affinity DataIC50: 2.66E+3nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166066BDBM50166066(CHEMBL362991 | Tyr-Pro-Phe-Pro-NH2 | [D-Pro4]morph...)
Affinity DataIC50: 3.69E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456334BDBM50456334(CHEMBL2371340)
Affinity DataIC50: 4.81E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456333BDBM50456333(CHEMBL2371361)
Affinity DataIC50: 2.69E+4nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456333BDBM50456333(CHEMBL2371361)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456338BDBM50456338(CHEMBL2371337)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456339BDBM50456339(CHEMBL2371336)
Affinity DataIC50: 5.65E+5nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50456338BDBM50456338(CHEMBL2371337)
Affinity DataIC50: 1.00E+6nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed