Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50036433
TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052309(Acetic acid (4R,5R)-7-chloro-1-dimethylaminomethyl...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052310(Acetic acid (4R,5R)-1-dimethylaminomethyl-5-(4-met...)
Affinity DataKi:  63nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052314(Acetic acid (4R,5R)-9-chloro-1-dimethylaminomethyl...)
Affinity DataKi:  569nMAssay Description:Inhibition of [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  1.40nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  2nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041505(CHEMBL33096 | Dimethyl-carbamic acid 5-(4-methoxy-...)
Affinity DataIC50:  9nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50052311(Acetic acid (4R,5R)-7-chloro-1-dimethylaminomethyl...)
Affinity DataIC50:  12nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50029417(CHEMBL277363 | [4-(4-Methoxy-phenyl)-4H-benzo[b]py...)
Affinity DataIC50:  17nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041506(Acetic acid 7-chloro-5-(4-methoxy-phenyl)-6-thia-1...)
Affinity DataIC50:  20nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041493(Acetic acid 5-phenyl-6-thia-10b-aza-benzo[e]azulen...)
Affinity DataIC50:  20nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041504(Butyric acid 5-phenyl-6-thia-10b-aza-benzo[e]azule...)
Affinity DataIC50:  22nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041513(CHEMBL416214 | Hexanoic acid 5-phenyl-6-thia-10b-a...)
Affinity DataIC50:  23nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041496(Butyric acid 5-(4-methoxy-phenyl)-6-thia-10b-aza-b...)
Affinity DataIC50:  28nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041502(Acetic acid 5-(4-methoxy-phenyl)-6-thia-10b-aza-be...)
Affinity DataIC50:  34nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  39nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041508(CHEMBL416040 | Pentanoic acid 5-phenyl-6-thia-10b-...)
Affinity DataIC50:  48nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50004704((+)-cis-Diltiazem | (2S,3S)-5-(2-(dimethylamino)et...)
Affinity DataIC50:  54nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052317(Acetic acid (4R,5R)-1-dimethylaminomethyl-5-phenyl...)
Affinity DataIC50:  139nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041485(Acetic acid 9-chloro-5-phenyl-6-thia-10b-aza-benzo...)
Affinity DataIC50:  150nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50041496(Butyric acid 5-(4-methoxy-phenyl)-6-thia-10b-aza-b...)
Affinity DataIC50:  150nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50041493(Acetic acid 5-phenyl-6-thia-10b-aza-benzo[e]azulen...)
Affinity DataIC50:  220nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50041502(Acetic acid 5-(4-methoxy-phenyl)-6-thia-10b-aza-be...)
Affinity DataIC50:  340nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50041508(CHEMBL416040 | Pentanoic acid 5-phenyl-6-thia-10b-...)
Affinity DataIC50:  610nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50041490(Acetic acid 9-chloro-5-(4-methoxy-phenyl)-6-thia-1...)
Affinity DataIC50:  651nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50029417(CHEMBL277363 | [4-(4-Methoxy-phenyl)-4H-benzo[b]py...)
Affinity DataIC50: >2.00E+3nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052315(Acetic acid 9-chloro-1-dimethylaminomethyl-5-(4-me...)
Affinity DataIC50: >2.00E+3nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052316(Acetic acid 9-chloro-1-dimethylaminomethyl-5-pheny...)
Affinity DataIC50: >2.00E+3nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052318(Acetic acid 1-dimethylaminomethyl-5-phenyl-6-thia-...)
Affinity DataIC50: >2.00E+3nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTranslocator protein(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50052312(Acetic acid (4R,5R)-1-dimethylaminomethyl-5-phenyl...)
Affinity DataIC50:  2.41E+3nMAssay Description:Ability to inhibit [3H]-PK 11195 binding to peripheral-type benzodiazepine receptor(PBR) in rat cerebral cortex homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed