Compile Data Set for Download or QSAR
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Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50022835
TargetFibroblast growth factor receptor 1(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50065306(3-[4-(1-formylpiperazin-4-yl)benzylidenyl]-2-indol...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of FGFR1K (unknown origin) autophosphorylation activity assessed as [32P] incorporationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Mouse)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM4882((Z)-3-[(3-(2-Carboxyethyl)-4-methylpyrrol-2-yl)met...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of acidic FGF-stimulated FGFR1 tyrosine autophosphorylation in mouse NIH/3T3 cells by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetFibroblast growth factor receptor 1(Human)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM4882((Z)-3-[(3-(2-Carboxyethyl)-4-methylpyrrol-2-yl)met...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of FGFR1K (unknown origin) autophosphorylation activity assessed as [32P] incorporationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB
PDB3D3D Structure (crystal)

TargetFibroblast growth factor receptor 1(Mouse)
New York University Medical Center

Curated by ChEMBL
LigandPNGBDBM50065306(3-[4-(1-formylpiperazin-4-yl)benzylidenyl]-2-indol...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of acidic FGF-stimulated FGFR1 tyrosine autophosphorylation in mouse NIH/3T3 cells by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed