Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50036518
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.510nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 22.4nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataIC50: 264nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataIC50: 557nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory concentration against human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.580nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataEC50: 2.61nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 136nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6.08nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.720nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 89nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0400nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.240nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6.10nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 3 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 269nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Human)
University of Michigan Medical Center
Curated by ChEMBL
University of Michigan Medical Center
Curated by ChEMBL
Affinity DataEC50: 0.190nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair