Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50007736
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066991((R)-2-(2-Benzyloxycarbonylamino-4-methyl-pentanoyl...)
Affinity DataIC50:  7nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066994((1-{(R)-1-[Bis-(4-chloro-phenyl)-phosphinoanecarbo...)
Affinity DataIC50:  350nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066989(CHEMBL127322 | [(R)-2-(2-Benzyloxycarbonylamino-4-...)
Affinity DataIC50:  370nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066993(CHEMBL127716 | [(R)-2-(2-Benzyloxycarbonylamino-4-...)
Affinity DataIC50:  430nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066990((R)-2-(2-Benzyloxycarbonylamino-4-methyl-pentanoyl...)
Affinity DataIC50:  600nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066987(CHEMBL127408 | [(R)-2-(2-Benzyloxycarbonylamino-4-...)
Affinity DataIC50:  5.20E+3nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066992(CHEMBL340840 | [(R)-2-(2-Benzyloxycarbonylamino-3-...)
Affinity DataIC50:  6.00E+3nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066986(CHEMBL127630 | [(R)-2-(2-Benzyloxycarbonylamino-3-...)
Affinity DataIC50:  7.40E+3nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066985(CHEMBL338195 | {1-[(R)-1-(Dimethyl-phosphinoanecar...)
Affinity DataIC50: >1.00E+4nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066995(CHEMBL126585 | [(R)-2-(2-Benzyloxycarbonylamino-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50066988(CHEMBL338878 | [(R)-2-(2-Benzyloxycarbonylamino-3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:inhibitory activity measured against recombinant human Calpain-I receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed