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Found 12 Enz. Inhib. hit(s) with all data for entry = 50034963
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057499((R)-8-Chloro-4,10b-dimethyl-1,4,4a,5,6,10b-hexahyd...)
Affinity DataKi:  9nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057501((S)-7-Chloro-4a-methyl-3,4,4a,9-tetrahydro-phenant...)
Affinity DataKi:  260nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072190((R)-8-Chloro-4,10b-dimethyl-1,5,6,10b-tetrahydro-2...)
Affinity DataKi:  920nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057499((R)-8-Chloro-4,10b-dimethyl-1,4,4a,5,6,10b-hexahyd...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50057501((S)-7-Chloro-4a-methyl-3,4,4a,9-tetrahydro-phenant...)
Affinity DataKi:  1.20E+3nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072190((R)-8-Chloro-4,10b-dimethyl-1,5,6,10b-tetrahydro-2...)
Affinity DataKi:  2.00E+4nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  1.20nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 2 receptor from human prostate homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072189((7aS,8R)-7a-Methyl-2-oxo-2,3,4,7,7a,8,9,10,10a,10b...)
Affinity DataIC50:  122nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 2 receptor from human prostate homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072189((7aS,8R)-7a-Methyl-2-oxo-2,3,4,7,7a,8,9,10,10a,10b...)
Affinity DataIC50:  127nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1 from recombinant CHO cells; No inhibition up to 10 uM concentrati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072191(1,2,5,6-Tetrahydro-pyrido[1,2-a]quinolin-3-one | 1...)
Affinity DataIC50:  298nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1 from recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50:  911nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1 from recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072192(3,4,5,6-Tetrahydrobenzo[c]quinolizin-3-(4aH)-one |...)
Affinity DataIC50:  5.13E+3nMAssay Description:Compound was evaluated for the inhibition of human Steroid 5-alpha-reductase type 1 from recombinant CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed