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Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50008394
TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073029(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-spiro[1,2,3,4-t...)
Affinity DataEC50:  66nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)
Affinity DataEC50:  10nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073031(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[1-oxospiro[2,3...)
Affinity DataEC50:  42nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataEC50:  1.30nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073032(1N-[2-(5-hydroxy-1,3,4,4a,5,10a-hexahydro-2H-chrom...)
Affinity DataEC50:  16nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073033(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[4-oxospiro[3,4...)
Affinity DataEC50:  1.80nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049481((R)-N-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)meth...)
Affinity DataEC50:  60nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073034(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-spiro[3,4-dihyd...)
Affinity DataEC50:  2.90nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073035(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[4-oxospiro[3,4...)
Affinity DataEC50:  37nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073036(1N-[2-[4-hydroxyspiro[3,4-dihydro-2H-chromene-2,3'...)
Affinity DataEC50:  1.20nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50066103(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[4-oxo-(2'S)-sp...)
Affinity DataEC50:  57nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073038(1N-[2-[1-hydroxyspiro[2,3-dihydro-1H-indene-2,4'-(...)
Affinity DataEC50:  19nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073040(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-spiro[2,3-dihyd...)
Affinity DataEC50:  60nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073039(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-spiro[2,3-dihyd...)
Affinity DataEC50:  630nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073042(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[1-oxospiro[2,3...)
Affinity DataEC50:  20nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073041(1N-[2-(1,3,4,4a,5,10a-hexahydro-2H-chromeno[2,3-c]...)
Affinity DataEC50:  25nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50069108(1-{[(2R)-1-{2,3-dihydrospiro[indene-1,4'-piperidin...)
Affinity DataEC50:  14nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073043(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-[4-oxo-(2'R)-sp...)
Affinity DataEC50:  1.20nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGrowth hormone secretagogue receptor type 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50073030(1N-[1-(1H-3-indolylmethyl)-2-oxo-2-spiro[2,3-dihyd...)
Affinity DataEC50:  37nMAssay Description:In vitro growth hormone release was determined in rat pituitary cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed