Compile Data Set for Download or QSAR
Report error Found 246 Enz. Inhib. hit(s) with all data for entry = 599
TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281282BDBM281282(US10022354, Example 222)
Affinity DataIC50: 0.0250nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281250BDBM281250(US10022354, Example 190)
Affinity DataIC50: 0.0370nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281249BDBM281249(US10022354, Example 189)
Affinity DataIC50: 0.0380nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281103BDBM281103(US10022354, Example 43)
Affinity DataIC50: 0.0390nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281279BDBM281279(US10022354, Example 219)
Affinity DataIC50: 0.0460nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281189BDBM281189(US10022354, Example 129)
Affinity DataIC50: 0.0470nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281089BDBM281089(US10022354, Example 29)
Affinity DataIC50: 0.0490nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281278BDBM281278(US10022354, Example 218)
Affinity DataIC50: 0.0500nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281101BDBM281101(US10022354, Example 41)
Affinity DataIC50: 0.0510nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281281BDBM281281(US10022354, Example 221)
Affinity DataIC50: 0.0510nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281180BDBM281180(US10022354, Example 120)
Affinity DataIC50: 0.0530nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281196BDBM281196(US10022354, Example 136)
Affinity DataIC50: 0.0540nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281100BDBM281100(US10022354, Example 40)
Affinity DataIC50: 0.0580nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281094BDBM281094(US10022354, Example 34)
Affinity DataIC50: 0.0580nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281188BDBM281188(US10022354, Example 128)
Affinity DataIC50: 0.0590nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281211BDBM281211(US10022354, Example 151)
Affinity DataIC50: 0.0650nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281240BDBM281240(US10022354, Example 180)
Affinity DataIC50: 0.0650nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281181BDBM281181(US10022354, Example 121)
Affinity DataIC50: 0.0660nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281172BDBM281172(US10022354, Example 112)
Affinity DataIC50: 0.0660nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281194BDBM281194(US10022354, Example 134)
Affinity DataIC50: 0.0710nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281218BDBM281218(US10022354, Example 158)
Affinity DataIC50: 0.0730nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281216BDBM281216(US10022354, Example 156)
Affinity DataIC50: 0.0740nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281284BDBM281284(US10022354, Example 224)
Affinity DataIC50: 0.0740nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281215BDBM281215(US10022354, Example 155)
Affinity DataIC50: 0.0750nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281195BDBM281195(US10022354, Example 135)
Affinity DataIC50: 0.0760nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281177BDBM281177(US10022354, Example 117)
Affinity DataIC50: 0.0770nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281243BDBM281243(US10022354, Example 183)
Affinity DataIC50: 0.0780nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281237BDBM281237(US10022354, Example 177)
Affinity DataIC50: 0.0780nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281288BDBM281288(US10022354, Example 228)
Affinity DataIC50: 0.0780nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281238BDBM281238(US10022354, Example 178)
Affinity DataIC50: 0.0800nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281102BDBM281102(US10022354, Example 42)
Affinity DataIC50: 0.0820nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281212BDBM281212(US10022354, Example 152)
Affinity DataIC50: 0.0830nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281095BDBM281095(US10022354, Example 35)
Affinity DataIC50: 0.0830nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281093BDBM281093(US10022354, Example 33)
Affinity DataIC50: 0.0870nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281261BDBM281261(US10022354, Example 201)
Affinity DataIC50: 0.0920nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281073BDBM281073(US10022354, Example 13)
Affinity DataIC50: 0.0940nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281210BDBM281210(US10022354, Example 150)
Affinity DataIC50: 0.0980nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281245BDBM281245(US10022354, Example 185)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281285BDBM281285(US10022354, Example 225)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281256BDBM281256(US10022354, Example 196)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281129BDBM281129(US10022354, Example 69)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281225BDBM281225(US10022354, Example 165)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281289BDBM281289(US10022354, Example 229)
Affinity DataIC50: 0.110nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281082BDBM281082(US10022354, Example 22)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281213BDBM281213(US10022354, Example 153)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281121BDBM281121(US10022354, Example 61)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281219BDBM281219(US10022354, Example 159)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281192BDBM281192(US10022354, Example 132)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281272BDBM281272(US10022354, Example 212)
Affinity DataIC50: 0.120nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

TargetLysine-specific demethylase 5A(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 281067BDBM281067(US10022354, Example 7)
Affinity DataIC50: 0.130nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details
US Patent

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