Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 978
TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 35667BDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataEC50:  40nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301711BDBM301711(US10131692, Compound 43 ([Val4]dDAVP))
Affinity DataEC50:  50nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301678BDBM301678(US10131692, Compound 10)
Affinity DataEC50:  70nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301674BDBM301674(US10131692, Compound 6)
Affinity DataEC50:  80nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301693BDBM301693(US10131692, Compound 25)
Affinity DataEC50:  80nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301699BDBM301699(US10131692, Compound 31)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301691BDBM301691(US10131692, Compound 23)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301676BDBM301676(US10131692, Compound 8)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301701BDBM301701(US10131692, Compound 33)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301669BDBM301669(US10131692, Compound 1)
Affinity DataEC50:  100nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301702BDBM301702(US10131692, Compound 34)
Affinity DataEC50:  110nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301708BDBM301708(US10131692, Compound 40)
Affinity DataEC50:  120nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301690BDBM301690(US10131692, Compound 22)
Affinity DataEC50:  140nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301704BDBM301704(US10131692, Compound 36)
Affinity DataEC50:  170nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301681BDBM301681(US10131692, Compound 13)
Affinity DataEC50:  190nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301698BDBM301698(US10131692, Compound 30)
Affinity DataEC50:  190nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301677BDBM301677(US10131692, Compound 9)
Affinity DataEC50:  190nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301684BDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  200nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301680BDBM301680(US10131692, Compound 12)
Affinity DataEC50:  210nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301703BDBM301703(US10131692, Compound 35)
Affinity DataEC50:  210nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301673BDBM301673(US10131692, Compound 5)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301709BDBM301709(US10131692, Compound 41)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 50205308BDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301686BDBM301686(US10131692, Compound 18)
Affinity DataEC50:  220nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301684BDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  230nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301679BDBM301679(US10131692, Compound 11)
Affinity DataEC50:  230nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301689BDBM301689(US10131692, Compound 21)
Affinity DataEC50:  250nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301706BDBM301706(US10131692, Compound 38)
Affinity DataEC50:  260nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301682BDBM301682(US10131692, Compound 14)
Affinity DataEC50:  260nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301688BDBM301688(US10131692, Compound 20)
Affinity DataEC50:  270nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301694BDBM301694(US10131692, Compound 26)
Affinity DataEC50:  270nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301700BDBM301700(US10131692, Compound 32)
Affinity DataEC50:  290nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301671BDBM301671(US10131692, Compound 3)
Affinity DataEC50:  290nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301687BDBM301687(US10131692, Compound 19)
Affinity DataEC50:  290nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301705BDBM301705(US10131692, Compound 37)
Affinity DataEC50:  300nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301707BDBM301707(US10131692, Compound 39)
Affinity DataEC50:  310nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301675BDBM301675(US10131692, Compound 7)
Affinity DataEC50:  310nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301696BDBM301696(US10131692, Compound 28)
Affinity DataEC50:  320nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301672BDBM301672(US10131692, Compound 4)
Affinity DataEC50:  330nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301692BDBM301692(US10131692, Compound 24)
Affinity DataEC50:  350nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301685BDBM301685(US10131692, Compound 17)
Affinity DataEC50:  350nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301697BDBM301697(US10131692, Compound 29)
Affinity DataEC50:  380nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301670BDBM301670(US10131692, Compound 2)
Affinity DataEC50:  390nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V2 receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301683BDBM301683(US10131692, Compound 15)
Affinity DataEC50:  450nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 35667BDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataEC50:  5.40E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 50205308BDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  6.59E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301711BDBM301711(US10131692, Compound 43 ([Val4]dDAVP))
Affinity DataEC50:  2.41E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301702BDBM301702(US10131692, Compound 34)
Affinity DataEC50:  4.02E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301694BDBM301694(US10131692, Compound 26)
Affinity DataEC50:  4.58E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandChemical structure of BindingDB Monomer ID 301674BDBM301674(US10131692, Compound 6)
Affinity DataEC50:  5.76E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

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