Compile Data Set for Download or QSAR
Report error Found 229 Enz. Inhib. hit(s) with all data for entry = 1033
LigandChemical structure of BindingDB Monomer ID 304006BDBM304006(US10138242, Compound 95)
Affinity DataIC50: 140nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304008BDBM304008(US10138242, Compound 97)
Affinity DataIC50: 160nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304005BDBM304005(US10138242, Compound 94)
Affinity DataIC50: 220nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303951BDBM303951(US10138242, Compound 37)
Affinity DataIC50: 240nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304007BDBM304007(US10138242, Compound 96)
Affinity DataIC50: 250nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304009BDBM304009(US10138242, Compound 98)
Affinity DataIC50: 300nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304010BDBM304010(US10138242, Compound 99)
Affinity DataIC50: 300nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304012BDBM304012(US10138242, Compound 101)
Affinity DataIC50: 420nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304011BDBM304011(US10138242, Compound 100)
Affinity DataIC50: 570nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304015BDBM304015(US10138242, Compound 104)
Affinity DataIC50: 620nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304013BDBM304013(US10138242, Compound 102)
Affinity DataIC50: 850nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303952BDBM303952(US10138242, Compound 38)
Affinity DataIC50: 880nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304014BDBM304014(US10138242, Compound 103)
Affinity DataIC50: 980nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303927BDBM303927(US10138242, Compound 13)
Affinity DataIC50: 990nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303974BDBM303974(US10138242, Compound 60)
Affinity DataIC50: 1.02E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303929BDBM303929(US10138242, Compound 15)
Affinity DataIC50: 1.09E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303919BDBM303919(US10138242, Compound 5)
Affinity DataIC50: 1.11E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303950BDBM303950(US10138242, Compound 36)
Affinity DataIC50: 1.12E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303930BDBM303930(US10138242, Compound 16)
Affinity DataIC50: 1.22E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303958BDBM303958(US10138242, Compound 44)
Affinity DataIC50: 1.27E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304016BDBM304016(US10138242, Compound 105)
Affinity DataIC50: 1.27E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304005BDBM304005(US10138242, Compound 94)
Affinity DataEC50:  1.40E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303953BDBM303953(US10138242, Compound 39)
Affinity DataIC50: 1.50E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303925BDBM303925(US10138242, Compound 11)
Affinity DataIC50: 1.70E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304006BDBM304006(US10138242, Compound 95)
Affinity DataEC50:  1.75E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304007BDBM304007(US10138242, Compound 96)
Affinity DataEC50:  1.92E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304008BDBM304008(US10138242, Compound 97)
Affinity DataEC50:  1.98E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303932BDBM303932(US10138242, Compound 18)
Affinity DataIC50: 2.00E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303949BDBM303949(US10138242, Compound 35)
Affinity DataIC50: 2.17E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303920BDBM303920(US10138242, Compound 6)
Affinity DataIC50: 2.27E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304009BDBM304009(US10138242, Compound 98)
Affinity DataEC50:  2.27E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303957BDBM303957(US10138242, Compound 43)
Affinity DataIC50: 2.38E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303966BDBM303966(US10138242, Compound 52)
Affinity DataIC50: 2.50E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304017BDBM304017(US10138242, Compound 106)
Affinity DataIC50: 2.50E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303928BDBM303928(US10138242, Compound 14)
Affinity DataIC50: 2.59E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303945BDBM303945(US10138242, Compound 31)
Affinity DataIC50: 2.62E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303935BDBM303935(US10138242, Compound 21)
Affinity DataIC50: 2.63E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304019BDBM304019(US10138242, Compound 108)
Affinity DataIC50: 2.70E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304010BDBM304010(US10138242, Compound 99)
Affinity DataEC50:  2.73E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303994BDBM303994(US10138242, Compound 80)
Affinity DataIC50: 2.76E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303964BDBM303964(US10138242, Compound 50)
Affinity DataIC50: 2.89E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303975BDBM303975(US10138242, Compound 61)
Affinity DataIC50: 2.96E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303962BDBM303962(US10138242, Compound 48)
Affinity DataIC50: 2.99E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304020BDBM304020(US10138242, Compound 109)
Affinity DataIC50: 3.30E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303944BDBM303944(US10138242, Compound 30)
Affinity DataIC50: 3.36E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303931BDBM303931(US10138242, Compound 17)
Affinity DataIC50: 3.41E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 304012BDBM304012(US10138242, Compound 101)
Affinity DataEC50:  3.44E+3nMAssay Description:The assay uses two types of beads: donor beads are coupled with streptavidin, and acceptor beads are coupled with an anti His-tag antibody. Upon exci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303948BDBM303948(US10138242, Compound 34)
Affinity DataIC50: 3.49E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303955BDBM303955(US10138242, Compound 41)
Affinity DataIC50: 3.75E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 303965BDBM303965(US10138242, Compound 51)
Affinity DataIC50: 4.00E+3nMAssay Description:Antitrypanosomal activity was tested on T. brucei brucei bloodstream from parasites (strain Lister 427, VATMITat 1.2). Stock solutions of compounds (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2019
Entry Details
US Patent

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