Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 3228
TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394383(US10308605, Example 30 | N-methyl-1-[1-(phenylsulf...)
Affinity DataIC50: 4.20nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394395(US10308605, Example 225 | 1-[5-(2,4-Difluorophenyl...)
Affinity DataIC50: 8.90nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394391(US10308605, Example 165 | 1-{5-(2-Fluorophenyl)-1-...)
Affinity DataIC50: 9nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394389(US10308605, Example 157 | Ethyl 1-(pyridazin-3-yls...)
Affinity DataIC50: 13nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394392(US10308605, Example 166 | 1-[5-(2-Fluorophenyl)-1-...)
Affinity DataIC50: 22nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394388(US10308605, Example 152 | 1-[1-(1-Benzothien-2-yls...)
Affinity DataIC50: 33nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394394(US10308605, Example 220 | N-Methyl-1-[5-(2-methylp...)
Affinity DataIC50: 36nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394386(US10308605, Example 43 | N-Methyl-1-[5-phenyl-1-(3...)
Affinity DataIC50: 51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394378(US10308605, Example 11 | Ethyl 1-[(4-methoxyphenyl...)
Affinity DataIC50: 51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394390(US10308605, Example 161 | 1-[5-(2-Fluorophenyl)-1-...)
Affinity DataIC50: 62nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394387(US10308605, Example 140)
Affinity DataIC50: 78nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394393(US10308605, Example 204 | N-Methyl-3-({4-[(methyla...)
Affinity DataIC50: 86nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394377(US10308605, Example 7 | N-Methyl-1-{5-(3-methylphe...)
Affinity DataIC50: 91nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent

TargetPotassium-transporting ATPase alpha chain 1(Pig)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394382(US10308605, Example 12 | 1-[(4-Methoxyphenyl)sulfo...)
Affinity DataIC50: 710nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/15/2020
Entry Details
US Patent