Compile Data Set for Download or QSAR
Report error Found 172 Enz. Inhib. hit(s) with all data for entry = 9071
TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438928(US10604489, Compound 89)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438926(US10604489, Compound 87 | US11180455, Compound 89)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438920(4-((1R,5S,9r)-9-methoxy-3-(2-oxaspiro[3.3]heptan-6...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438916(4-((1R,5S,9r)-9-methoxy-3-(spiro[3.3]heptan-2-yl)-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438943(US10604489, Compound 104 | US11180455, Compound 10...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438945(tert-butyl (3-phenylbicyclo[1.1.1]pentan-1-yl)carb...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438939(4-((1R,5S,9r)-3-((1H-pyrazol-5-yl)methyl)-9-methox...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438941(US10604489, Compound 102 | US11180455, Compound 10...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438936(5-((1R,5S,9r)-3-(2-(1,1-dioxidoisothiazolidin-2-yl...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438935(4-((1R,5S,9r)-3-((1H-imidazol-5-yl)methyl)-9-metho...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438933(US10604489, Compound 94 | US11180455, Compound 94)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438958(4-((1R,5S,9r)-3-((1H-indol-2-yl)methyl)-9-methoxy-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438948(US10604489, Compound 109 | US11180455, Compound 10...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438844(3-((1R,5S,9r)-3-(4,4-difluorocyclohexyl)-9-methoxy...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438978(US10604489, Compound 139 | US11180455, Compound 13...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438846(3-((1R,5S,9r)-3-(bicyclo[3.1.0]hexan-3-yl)-9-metho...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438977(3-((1R,5S,9r)-3-(2-cyclopropylethyl)-9-methoxy-3-a...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438972(3-((1R,5S,9r)-9-methoxy-3-(2-oxaspiro[3.3]heptan-6...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438839(3-((1R,5S,9r)-9-methoxy-3-(2-oxaspiro[3.5]nonan-7-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438973(4-((1R,5S,9S)-9-methoxy-3-((S)-pentan-2-yl)-3-azab...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438841(3-((1R,5S,9r)-9-methoxy-3-(7-oxaspiro[3.5]nonan-2-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438968(3-((1R,5S,9r)-9-methoxy-3-(spiro[3.3]heptan-2-yl)-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438967(3-((1R,5S,9r)-9-methoxy-3-(2-methoxyethyl)-3-azabi...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438838(US10604489, Compound 2 | US11180455, Compound 2)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438969(US10604489, Compound 130 | US11180455, Compound 13...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438965(4-((1R,5S,9r)-3-((1H-indol-3-yl)methyl)-9-methoxy-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438992(3-((1R,5S,9r)-3-(but-3-yn-1-yl)-9-methoxy-3-azabic...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438863(3-((1R,5S,9r)-3-isopropyl-9-methoxy-3-azabicyclo[3...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438991(3-((1R,5S,9r)-3-((1H-indazol-3-yl)methyl)-9-methox...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438862(3-((1R,5S,9r)-9-methoxy-3-phenethyl-3-azabicyclo[3...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438994(3-((1R,5S,9r)-3-(3-fluoropropyl)-9-methoxy-3-azabi...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438993(US10604489, Compound 156 | US11180455, Compound 15...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438864(3-benzyl-1,5,3-dioxazepane | US10604489, Compound ...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438988(3-((1R,5S,9r)-9-methoxy-3-(1-phenylazetidin-3-yl)-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438858(3-((1R,5S,9r)-3-benzyl-9-methoxy-3-azabicyclo[3.3....)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438990(4-((1R,5S,9r)-9-methoxy-3-((5-methyl-1H-imidazol-2...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438861(US10604489, Compound 54 | 3-((1R,5S,9r)-9-methoxy-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438989(US10604489, Compound 152 | US11180455, Compound 15...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438859(3-((1R,5S,9r)-9-methoxy-3-azabicyclo[3.3.1]nonan-9...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438853(3-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438983(4-((1R,5S,9s)-9-methoxy-3-((1S,2S)-2-methylcyclobu...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438852(US10604489, Compound 16)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438986(3-((1R,5S,9r)-9-methoxy-34(2-methyl-1H-imidazol-4-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438855(US10604489, Compound 19 | US11180455, Compound 19)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438985(US10604489, Compound 148 | US11180455, Compound 14...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438854(4-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438980(US10604489, Compound 141 | US11180455, Compound 14...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438849(4-((1R,5S,9r)-9-methoxy-3-(7-oxaspiro[3.5]nonan-2-...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438979(US10604489, Compound 140 | US11180455, Compound 14...)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Alkermes

US Patent
LigandPNGBDBM438848(US10604489, Compound 12)
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

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