Compile Data Set for Download or QSAR
Report error Found 119 Enz. Inhib. hit(s) with all data for entry = 9588
TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476189BDBM476189(US10865384, Example 2l | US10865384, Compound IM-3...)
Affinity DataIC50: 2.70nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476192BDBM476192(US10865384, Example 2o | US10865384, Compound IM-3...)
Affinity DataIC50: 2.80nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476187BDBM476187(US10865384, Example 2j | US10865384, Compound IM-3...)
Affinity DataIC50: 3.20nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476188BDBM476188(US10865384, Example 2k | US10865384, Compound IM-3...)
Affinity DataIC50: 3.30nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476190BDBM476190(US10865384, Example 2m | US10865384, Compound IM-4...)
Affinity DataIC50: 3.70nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491733BDBM50491733(CHEMBL2385554 | US10865384, Compound IM-26)
Affinity DataIC50: 4.30nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476191BDBM476191(US10865384, Example 2n | US10865384, Compound IM-3...)
Affinity DataIC50: 4.40nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491730BDBM50491730(CHEMBL2385555 | US10865384, Compound IM-19)
Affinity DataIC50: 4.70nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476185BDBM476185(US10865384, Example 2h | US10865384, Compound IM-3...)
Affinity DataIC50: 5nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476186BDBM476186(US10865384, Example 2i | US10865384, Compound IM-3...)
Affinity DataIC50: 5.30nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476175BDBM476175(US10865384, Example 1a | US10865384, Compound IM-3...)
Affinity DataIC50: 6.40nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476175BDBM476175(US10865384, Example 1a | US10865384, Compound IM-3...)
Affinity DataIC50: 6.40nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476175BDBM476175(US10865384, Example 1a | US10865384, Compound IM-3...)
Affinity DataIC50: 6.70nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476175BDBM476175(US10865384, Example 1a | US10865384, Compound IM-3...)
Affinity DataIC50: 6.80nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476175BDBM476175(US10865384, Example 1a | US10865384, Compound IM-3...)
Affinity DataIC50: 6.80nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491729BDBM50491729(CHEMBL2385556 | US10865384, Compound IM-27)
Affinity DataIC50: 8.40nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476184BDBM476184(US10865384, Example 2g | US10865384, Compound IM-3...)
Affinity DataIC50: 9.5nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476196BDBM476196(US10865384, Example 2s | US10865384, Compound IM-4...)
Affinity DataIC50: 11nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476205BDBM476205(US10865384, Example 4b | US10865384, Compound IM-1...)
Affinity DataIC50: 14nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476177BDBM476177(US10865384, Example 1c | US10865384, Compound IM-2...)
Affinity DataIC50: 15nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476177BDBM476177(US10865384, Example 1c | US10865384, Compound IM-2...)
Affinity DataIC50: 15nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476177BDBM476177(US10865384, Example 1c | US10865384, Compound IM-2...)
Affinity DataIC50: 16nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476177BDBM476177(US10865384, Example 1c | US10865384, Compound IM-2...)
Affinity DataIC50: 16nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476206BDBM476206(US10865384, Example 4c | US10865384, Compound IM-1...)
Affinity DataIC50: 19nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476176BDBM476176(US10865384, Example 1b | US10865384, Compound IM-3...)
Affinity DataIC50: 20nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491728BDBM50491728(CHEMBL2385557 | US10865384, Compound IM-4)
Affinity DataIC50: 20nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476207BDBM476207(US10865384, Example 4d | US10865384, Compound IM-1...)
Affinity DataIC50: 20nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50044784BDBM50044784(CHEBI:79090 | SB-202190 | US10865384, Compound SB2...)
Affinity DataIC50: 24nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192501BDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 24nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476182BDBM476182(US10865384, Example 2e | US10865384, Compound IM-2...)
Affinity DataIC50: 24nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476194BDBM476194(US10865384, Example 2q | US10865384, Compound IM-4...)
Affinity DataIC50: 26nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476176BDBM476176(US10865384, Example 1b | US10865384, Compound IM-3...)
Affinity DataIC50: 32nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476176BDBM476176(US10865384, Example 1b | US10865384, Compound IM-3...)
Affinity DataIC50: 32nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476176BDBM476176(US10865384, Example 1b | US10865384, Compound IM-3...)
Affinity DataIC50: 32nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476176BDBM476176(US10865384, Example 1b | US10865384, Compound IM-3...)
Affinity DataIC50: 32nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476208BDBM476208(US10865384, Example 4e | US10865384, Compound IM-1...)
Affinity DataIC50: 33nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192501BDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 43nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192501BDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 43nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476209BDBM476209(US10865384, Example 4f | US10865384, Compound IM-1...)
Affinity DataIC50: 43nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491733BDBM50491733(CHEMBL2385554 | US10865384, Compound IM-26)
Affinity DataIC50: 44nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50491733BDBM50491733(CHEMBL2385554 | US10865384, Compound IM-26)
Affinity DataIC50: 44nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476193BDBM476193(US10865384, Example 2p | US10865384, Compound IM-4...)
Affinity DataIC50: 45nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476195BDBM476195(US10865384, Example 2r | US10865384, Compound IM-4...)
Affinity DataIC50: 47nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50044784BDBM50044784(CHEBI:79090 | SB-202190 | US10865384, Compound SB2...)
Affinity DataIC50: 53nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform delta(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50044784BDBM50044784(CHEBI:79090 | SB-202190 | US10865384, Compound SB2...)
Affinity DataIC50: 53nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476199BDBM476199(US10865384, Example 3b | US10865384, Compound IM-2...)
Affinity DataIC50: 55nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192501BDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 63nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetCasein kinase I isoform epsilon(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 192501BDBM192501(US9187470, 104 (SB203580) | US10865384, Compound S...)
Affinity DataIC50: 63nMAssay Description:Table 3: Small molecules were tested for their inhibitory activities towards casein kinase 1 delta (CK1δ) and 1 epsilon (CK1ϵ). The in vit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476204BDBM476204(US10865384, Example 4a | US10865384, Compound IM-1...)
Affinity DataIC50: 73nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
Agency For Science, Technology and Research

US Patent
LigandChemical structure of BindingDB Monomer ID 476177BDBM476177(US10865384, Example 1c | US10865384, Compound IM-2...)
Affinity DataIC50: 73nMAssay Description:Table 2: The p38 MAPK IC50 values of selected compounds except IM-32 to IM-44 were determined using the HitHunter p38 MAP kinase binding assay from D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2021
Entry Details
US Patent

Displayed 1 to 50 (of 119 total ) | Next | Last >>
Jump to: