Compile Data Set for Download or QSAR
Report error Found 420 Enz. Inhib. hit(s) with all data for entry = 9964
LigandChemical structure of BindingDB Monomer ID 503879BDBM503879(1-[3-[4-[[8-amino-6-(4-methyl-3-pyridyl)- 2,7-naph...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503863BDBM503863(trans-N-[8-amino-6-(4-methyl-3-pyridyl)- 2,7-napht...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504044BDBM504044(US11034692, Compound 313)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503914BDBM503914((1S,2S)-N-(8-amino-5-fluoro-6-(4- methylpyridin-3-...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504062BDBM504062((1R,2R)-N-(8-amino-6-(4-methylpyridin- 3-yl)-2,7-n...)
Affinity DataKi: <0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504049BDBM504049((1R,2S)—N-(8-amino-5-cyclopropyl-6-(4-methylp...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504051BDBM504051((1S,2S)—N-(8-amino-6-(4-methyl-2-phenylpyridi...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503940BDBM503940(1-(3-(4-(8-amino-6-(4-methylpyridin-3- yl)-2,7-nap...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503988BDBM503988(2-[[8-amino-6-(4-methylpyridin-3-yl)-2,7- naphthyr...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503999BDBM503999(3-[[8-Amino-6-(4-methylpyridin-3-yl)-2,7- naphthyr...)
Affinity DataKi:  0.0210nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503978BDBM503978(US11034692, Compound 247)
Affinity DataKi:  0.0220nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504027BDBM504027((1S,2S)—N-[8-amino-6-(2,6-dichlorophenyl)-2,7...)
Affinity DataKi:  0.0260nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503943BDBM503943(1-(3-(8-amino-6-(4-methylpyridin-3-yl)- 2,7-naphth...)
Affinity DataKi:  0.0260nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503916BDBM503916((1S,2S)-N-(8-amino-6-(4-methylpyridin-3- yl)-2,7-n...)
Affinity DataKi:  0.0270nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504034BDBM504034((1R,2R)—N-(8-amino-6-(2-chloro-6-fluorophenyl...)
Affinity DataKi:  0.0270nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504050BDBM504050(US11034692, Compound 318)
Affinity DataKi:  0.0320nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504030BDBM504030((1R,2R)—N-[8-amino-6-(2-methylphenyl)-2,7-nap...)
Affinity DataKi:  0.0360nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503936BDBM503936(US11034692, Compound 214)
Affinity DataKi:  0.0390nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504023BDBM504023(US11034692, Compound 292)
Affinity DataKi:  0.0420nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503977BDBM503977((1S,2S)—N-(8-amino-6-(4-(2-hydroxyethyl)pyrid...)
Affinity DataKi:  0.0450nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503892BDBM503892(trans-N-(8-amino-5-chloro-6-(4- methylpyridin-3-yl...)
Affinity DataKi:  0.0470nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503926BDBM503926(trans-N-(8-amino-6-(4-methyl-2- phenylpyridin-3-yl...)
Affinity DataKi:  0.0510nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503939BDBM503939(2-(4-(8-amino-6-(4-methylpyridin-3-yl)- 2,7-naphth...)
Affinity DataKi:  0.0610nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503839BDBM503839(trans-N-[8-amino-6-(4-methyl-3-pyridyl)- 2,7-napht...)
Affinity DataKi:  0.0630nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504009BDBM504009((R)-2-(4-(8-amino-6-(4-methylpyridin-3- yl)-2,7-na...)
Affinity DataKi:  0.0680nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504041BDBM504041(US11034692, Compound 310)
Affinity DataKi:  0.0680nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504032BDBM504032((1R,2R)—N-[8-amino-6-(5-cyano-2-methylphenyl)...)
Affinity DataKi:  0.0690nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504058BDBM504058(US11034692, Compound 326)
Affinity DataKi:  0.0740nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504017BDBM504017((1R,2R)-N-[8-amino-6-(5-hydroxy-2- methylphenyl)-2...)
Affinity DataKi:  0.0780nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503960BDBM503960((1S,2S)—N-(8-amino-5-chloro-6-(4-methylpyridi...)
Affinity DataKi:  0.0780nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503925BDBM503925(trans-N-(8-amino-5-methyl-6-(4- methylpyridin-3-yl...)
Affinity DataKi:  0.0880nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503985BDBM503985(US11034692, Compound 253)
Affinity DataKi:  0.0890nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503795BDBM503795(3-(4-Ethylpyridin-3-yl)-N6-(1-piperidin-4- yl-1H-p...)
Affinity DataKi:  0.100nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504038BDBM504038((1S,2S)—N-[8-amino-6-(2,6-difluorophenyl)-2,7...)
Affinity DataKi:  0.112nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504003BDBM504003(trans-N-(8-amino-6-(5-fluoro-2- methylphenyl)-2,7-...)
Affinity DataKi:  0.113nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504060BDBM504060(US11034692, Compound 328)
Affinity DataKi:  0.114nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504006BDBM504006((1R,2S)—N-[8-amino-5-chloro-6-(4-methylpyridi...)
Affinity DataKi:  0.116nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504002BDBM504002(2-(4-[[8-amino-6-(4-methylpyridin-3-yl)- 2,7-napht...)
Affinity DataKi:  0.118nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504000BDBM504000((4-[[8-Amino-6-(4-methylpyridin-3-yl-2,7- naphthyr...)
Affinity DataKi:  0.134nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503874BDBM503874(US11034692, Compound 212 | trans-N-[8-amino-6-(4-m...)
Affinity DataKi:  0.135nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503945BDBM503945(cis-N-(8-amino-6-(3,4-dihydro-2H- pyrido[4,3-b][1,...)
Affinity DataKi:  0.135nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504008BDBM504008((1R,2S)—N-[8-amino-5-ethyl-6-(4-methylpyridin...)
Affinity DataKi:  0.139nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504004BDBM504004(trans-N-[8-amino-6-(5-hydroxy-2- methylphenyl)-2,7...)
Affinity DataKi:  0.147nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503869BDBM503869(trans-N-[8-amino-6-(4-methyl-3-pyridyl)- 2,7-napht...)
Affinity DataKi:  0.150nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504036BDBM504036((1S,2S)—N-[8-amino-6-(2-chlorophenyl)-2,7-nap...)
Affinity DataKi:  0.152nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503932BDBM503932(cis-N-(8-amino-6-(2,3-dihydro-1H- pyrrolo[2,3-c]py...)
Affinity DataKi:  0.154nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503956BDBM503956(trans-N-(8-amino-6-(4-methylpyridin-3- yl)-2,7-nap...)
Affinity DataKi:  0.173nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 503981BDBM503981((3R)-3-(4-[[8-amino-6-(4-methylpyridin-3-yl)-2,7-n...)
Affinity DataKi:  0.184nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504040BDBM504040((1S,2S)—N-[8-amino-6-[4-methyl-6-(1,3-oxazol-...)
Affinity DataKi:  0.184nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 504015BDBM504015((1S,2S,3R)—N-[8-amino-6-(4-methylpyridin-3-yl...)
Affinity DataKi:  0.188nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

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