Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 10067
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511679(4-(1-phenyl-1H-indazol-6- yl)pyridin-2-amine | US1...)
Affinity DataIC50:  1.17nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511678(4-(1-(m-tolyl)-1H-indazol-6- yl)pyridin-2-amine | ...)
Affinity DataIC50:  280nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511689(N-(1-(m-tolyl)-1H-indazol-6- yl)azetidine-3-carbox...)
Affinity DataIC50:  510nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511686(N-(azetidin-3-yl)-1-phenyl- 1H-indazole-6-carboxam...)
Affinity DataIC50:  580nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511683(4-(3-cyclopropyl-1-phenyl- 1H-indazol-6-yl)pyridin...)
Affinity DataIC50:  700nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511687(N-(piperidin-4-yl)-1-(m- tolyl)-1H-indazole-6- car...)
Affinity DataIC50:  790nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511690(US11083720, Compound C-72)
Affinity DataIC50:  1.20E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511688(1-phenyl-N-(piperidin-4-yl)- 1H-indazole-6-carboxa...)
Affinity DataIC50:  2.30E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKetohexokinase(Homo sapiens (Human))
Regents Of The University Of Colorado, A Body Corporate

US Patent
LigandPNGBDBM511684(N-(azetidin-3-yl)-1-(m-tolyl)- 1H-indazole-6-carbo...)
Affinity DataIC50:  2.30E+3nMAssay Description:Specific high-throughput screening assays were developed for KHK-C and KHK-A using recombinant proteins. Purified human recombinant KHK-C and KHK-A w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent