Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 10752
LigandChemical structure of BindingDB Monomer ID 563544BDBM563544(US11407768, Compound 1)
Affinity DataEC50:  0.0500nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563546BDBM563546(US11407768, Compound 3)
Affinity DataEC50:  0.0900nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563547BDBM563547(US11407768, Compound 4)
Affinity DataEC50:  0.100nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565695BDBM565695(US11407768, Compound 74)
Affinity DataEC50:  0.150nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565454BDBM565454(US11407768, Compound 53)
Affinity DataEC50:  0.230nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565696BDBM565696(US11407768, Compound 75)
Affinity DataEC50:  0.370nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563553BDBM563553(US11407768, Compound 10)
Affinity DataEC50:  0.400nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563495BDBM563495(US11407763, Example 45 | (2S)-2-amino-3-(4-(2- am...)
Affinity DataEC50:  0.460nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563556BDBM563556(US11407768, Compound 14)
Affinity DataEC50:  0.5nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563558BDBM563558(US11407768, Compound 29)
Affinity DataEC50:  0.560nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565456BDBM565456(US11407768, Compound 54)
Affinity DataEC50:  0.570nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563549BDBM563549(US11407768, Compound 6)
Affinity DataEC50:  0.620nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565561BDBM565561(US11407768, Compound 71)
Affinity DataEC50:  0.630nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563501BDBM563501(US11407768, Compound 22)
Affinity DataEC50:  0.630nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563503BDBM563503(US11407768, Compound 30 | (2S)-2-amino-3-(4-(2- am...)
Affinity DataEC50:  0.650nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565449BDBM565449(US11407768, Compound 51)
Affinity DataEC50:  0.720nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563504BDBM563504(US11407768, Compound 32)
Affinity DataEC50:  0.760nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565498BDBM565498(US11407768, Compound 65)
Affinity DataEC50:  0.770nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565503BDBM565503(US11407768, Compound 66)
Affinity DataEC50:  0.800nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565452BDBM565452(US11407768, Compound 52)
Affinity DataEC50:  0.810nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563563BDBM563563(US11407768, Compound 36)
Affinity DataEC50:  0.840nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563560BDBM563560(US11407768, Compound 31)
Affinity DataEC50:  0.850nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565483BDBM565483(US11407768, Compound 60)
Affinity DataEC50:  0.850nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565483BDBM565483(US11407768, Compound 60)
Affinity DataEC50:  0.850nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563548BDBM563548(US11407768, Compound 5)
Affinity DataEC50:  0.860nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565476BDBM565476(US11407768, Compound 57)
Affinity DataEC50:  0.890nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565506BDBM565506(US11407768, Compound 67)
Affinity DataEC50:  0.930nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565474BDBM565474(US11407768, Compound 56)
Affinity DataEC50:  0.930nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565478BDBM565478(US11407768, Compound 58)
Affinity DataEC50:  0.930nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563562BDBM563562(US11407768, Compound 33)
Affinity DataEC50:  0.960nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565481BDBM565481(US11407768, Compound 59)
Affinity DataEC50:  1.04nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563566BDBM563566(US11407768, Compound 40)
Affinity DataEC50:  1.08nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565494BDBM565494(US11407768, Compound 63)
Affinity DataEC50:  1.09nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563568BDBM563568(US11407768, Compound 48)
Affinity DataEC50:  1.16nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563550BDBM563550(US11407768, Compound 7)
Affinity DataEC50:  1.22nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565492BDBM565492(US11407768, Compound 62)
Affinity DataEC50:  1.30nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565694BDBM565694(US11407768, Compound 73)
Affinity DataEC50:  1.33nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565486BDBM565486(US11407768, Compound 61)
Affinity DataEC50:  1.36nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565693BDBM565693(US11407768, Compound 72)
Affinity DataEC50:  1.38nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563545BDBM563545(US11407768, Compound 2)
Affinity DataEC50:  1.40nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565496BDBM565496(US11407768, Compound 64)
Affinity DataEC50:  1.40nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565446BDBM565446(US11407768, Compound 50)
Affinity DataEC50:  1.46nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565530BDBM565530(US11407768, Compound 70)
Affinity DataEC50:  1.51nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563552BDBM563552(US11407768, Compound 9)
Affinity DataEC50:  1.61nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563540BDBM563540(US11407768, Compound 48)
Affinity DataEC50:  1.76nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563551BDBM563551(US11407768, Compound 8)
Affinity DataEC50:  1.78nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565528BDBM565528(US11407768, Compound 69)
Affinity DataEC50:  1.84nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 565470BDBM565470(US11407768, Compound 55)
Affinity DataEC50:  2.22nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563565BDBM563565(US11407768, Compound 38)
Affinity DataEC50:  2.40nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 563507BDBM563507(US11407768, Compound 37)
Affinity DataEC50:  3.60nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
11/5/2022
Entry Details
US Patent

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