Compile Data Set for Download or QSAR
maximum 50k data
Found 327 Enz. Inhib. hit(s) with all data for entry = 10831
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572127((R)-N-(4-(3-((6-fluoroquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572123((R)-N-(2-chloro-4-(3-(quinazolin-2- ylamino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572060((R)-N-(4-(3-((6-chloroquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572061((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572061((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572062((R)-N-(4-(3-(isoquinolin-3- ylamino)pyrrolidine-1-...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572063((R)-N-(4-(3-((6-fluoroquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572063((R)-N-(4-(3-((6-fluoroquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572066((R)-N-(4-(3-(pyrido[3,4-d]pyrimidin- 2-ylamino)pyr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572067((R)-N-(4-(3-((7-methylquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572068((R)-N-(4-(3-((7- (methylsulfonyl)quinazolin-2- yl)...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572068((R)-N-(4-(3-((7- (methylsulfonyl)quinazolin-2- yl)...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572069((R)-N-(4-(3-((7-methoxyquinazolin- 2-yl)amino)pyrr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572070((R)-N-(4-(3-((7-fluoroquinazolin-2- yl)amino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572072((R)-N-(4-(3-((7-cyanoquinazolin-2- yl)amino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572072((R)-N-(4-(3-((7-cyanoquinazolin-2- yl)amino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572073((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572073((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572074((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572074((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572075((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572075((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572076((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572077((R)-N-(4-(3-((7-oxo-7,8- dihydropyrido[2,3-d]pyrim...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572078((R)-N-(4-(3-((8-isopropyl-7-oxo-7,8- dihydropyrido...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572078((R)-N-(4-(3-((8-isopropyl-7-oxo-7,8- dihydropyrido...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572078((R)-N-(4-(3-((8-isopropyl-7-oxo-7,8- dihydropyrido...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572091((R)-2-((1-(4- propionamidobenzoyl)pyrrolidin-3- yl...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572091((R)-2-((1-(4- propionamidobenzoyl)pyrrolidin-3- yl...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572092((R)-2-((1-(4- propionamidobenzoyl)pyrrolidin-3- yl...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572092((R)-2-((1-(4- propionamidobenzoyl)pyrrolidin-3- yl...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572092((R)-2-((1-(4- propionamidobenzoyl)pyrrolidin-3- yl...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572075((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572075((R)-2-((1-(4- acrylamidobenzoyl)pyrrolidin-3- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572094((R)-N,N-dimethyl-2-((1-(4- propionamidobenzoyl)pyr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572094((R)-N,N-dimethyl-2-((1-(4- propionamidobenzoyl)pyr...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572095((R)-N-(4-(3-((7-oxo-7,8- dihydropyrido[2,3-d]pyrim...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572096((R)-N-(4-(3-((8-isopropyl-7-oxo-7,8- dihydropyrido...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572097((R)-N-(2-fluoro-4-(3-(quinazolin-2- ylamino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572097((R)-N-(2-fluoro-4-(3-(quinazolin-2- ylamino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572102((R)-N-(5-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572104((R)-N-(2-fluoro-4-(3-((6- fluoroquinazolin-2- yl)a...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572105((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572105((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572106((R)-N-(2-methoxy-4-(3-(quinazolin- 2-ylamino)pyrro...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572107((R)-N-(2-methyl-4-(3-(quinazolin-2- ylamino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572107((R)-N-(2-methyl-4-(3-(quinazolin-2- ylamino)pyrrol...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572112((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-K/Cyclin-dependent kinase 12(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572114((R)-1-(6-(3-(quinazolin-2- ylamino)pyrrolidine-1-c...)
Affinity DataIC50: <100nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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