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Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 10942
TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580132BDBM580132(US11498896, Compound 86)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580136BDBM580136(US11498896, Compound 98a)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50130293BDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580162BDBM580162(US11498896, Compound 211)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580141BDBM580141(US11498896, Compound 106)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580142BDBM580142(US11498896, Compound 110)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580148BDBM580148(US11498896, Compound 135)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580149BDBM580149(US11498896, Compound 137)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580146BDBM580146(US11498896, Compound 123)
Affinity DataKi: <100nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580152BDBM580152(US11498896, Compound 157)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580151BDBM580151(US11498896, Compound 144)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580157BDBM580157(US11498896, Compound 205)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50001884BDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580158BDBM580158(US11498896, Compound 206)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580155BDBM580155(US11498896, Compound 204b)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580161BDBM580161(US11498896, Compound 210)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580125BDBM580125(US11498896, Compound 27)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580159BDBM580159(US11498896, Compound 208)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580160BDBM580160(US11498896, Compound 209)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580130BDBM580130(US11498896, Compound 68)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50518039BDBM50518039(CHEMBL4467883 | US11498896, Compound 90)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580134BDBM580134(US11498896, Compound 91)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580131BDBM580131(US11498896, Compound 78)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580137BDBM580137(US11498896, Compound 99)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580140BDBM580140(US11498896, Compound 102a)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580135BDBM580135(US11498896, Compound 96)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580143BDBM580143(US11498896, Compound 112)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580145BDBM580145(US11498896, Compound 122)
Affinity DataKi:  550nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50518027BDBM50518027(CHEMBL4550815 | US11498896, Compound 1)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580154BDBM580154(US11498896, Compound 202b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580126BDBM580126(US11498896, Compound 54)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580124BDBM580124(US11498896, Compound 18b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580127BDBM580127(US11498896, Compound 55)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580147BDBM580147(US11498896, Compound 125)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580128BDBM580128(US11498896, Compound 59 | US11498896, Compound 59b)
Affinity DataKi:  5.50E+3nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580153BDBM580153(US11498896, Compound 164)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580150BDBM580150(US11498896, Compound 140)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580123BDBM580123(US11498896, Compound 7)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
The Broad Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 580128BDBM580128(US11498896, Compound 59 | US11498896, Compound 59b)
Affinity DataKi:  2.00E+4nMAssay Description:The D2 binding Ki values were determined using a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2023
Entry Details
US Patent