Compile Data Set for Download or QSAR
Report error Found 79 Enz. Inhib. hit(s) with all data for entry = 11550
TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626167(US11786528, Example 36)
Affinity DataIC50: 1.5nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626180(US11786528, Example 40)
Affinity DataIC50: 2nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625941(US11786528, Comparative Example 1)
Affinity DataIC50: 2.20nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626168(US11786528, Example 37)
Affinity DataIC50: 2.70nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626111(US11786528, Example 26)
Affinity DataIC50: 2.80nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626126(US11786528, Example 28)
Affinity DataIC50: 3.20nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626116(US11786528, Example 27)
Affinity DataIC50: 3.20nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625944(2-[(3-methylphenyl)methyl]-6-(1,2-thiazol-3-yl)-2H...)
Affinity DataIC50: 3.5nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626148(US11786528, Example 35)
Affinity DataIC50: 4.20nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626176(US11786528, Example 39)
Affinity DataIC50: 4.30nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626170(US11786528, Example 38)
Affinity DataIC50: 4.30nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625979(US11786528, Example 4)
Affinity DataIC50: 4.90nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626022(US11786528, Example 11)
Affinity DataIC50: 4.90nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626064(US11786528, Example 21)
Affinity DataIC50: 5nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626015(US11786528, Example 10)
Affinity DataIC50: 5.10nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626057(US11786528, Example 19)
Affinity DataIC50: 5.60nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626138(US11786528, Example 31)
Affinity DataIC50: 5.70nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625949(US11786528, Example 3 | US11786528, Example 2)
Affinity DataIC50: 6.70nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626028(US11786528, Example 12)
Affinity DataIC50: 7.90nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626100(US11786528, Example 24)
Affinity DataIC50: 7.90nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626134(US11786528, Example 30)
Affinity DataIC50: 8nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626039(US11786528, Example 16)
Affinity DataIC50: 8.30nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626143(US11786528, Example 32)
Affinity DataIC50: 10nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625997(US11786528, Example 8)
Affinity DataIC50: 11nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626195(US11786528, Example 43)
Affinity DataIC50: 13nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626059(US11786528, Example 20)
Affinity DataIC50: 13nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626035(US11786528, Example 14)
Affinity DataIC50: 14nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626133(US11786528, Example 29)
Affinity DataIC50: 15nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626034(US11786528, Example 13)
Affinity DataIC50: 15nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626198(US11786528, Example 44)
Affinity DataIC50: 15nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626046(US11786528, Example 18)
Affinity DataIC50: 18nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626108(US11786528, Example 25)
Affinity DataIC50: 18nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625994(US11786528, Example 7)
Affinity DataIC50: 24nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626144(US11786528, Example 33)
Affinity DataIC50: 27nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626076(US11786528, Example 22)
Affinity DataIC50: 27nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626077(US11786528, Example 23)
Affinity DataIC50: 29nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626205(US11786528, Example 45)
Affinity DataIC50: 31nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626206(US11786528, Example 46)
Affinity DataIC50: 37nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626006(US11786528, Example 9)
Affinity DataIC50: 41nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625949(US11786528, Example 3 | US11786528, Example 2)
Affinity DataIC50: 41nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625989(US11786528, Example 5)
Affinity DataIC50: 47nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626044(US11786528, Example 17)
Affinity DataIC50: 54nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626185(US11786528, Example 42)
Affinity DataIC50: 61nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626146(US11786528, Example 34)
Affinity DataIC50: 67nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Exscientia

US Patent
LigandPNGBDBM625941(US11786528, Comparative Example 1)
Affinity DataIC50: 114nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM625993(US11786528, Example 6)
Affinity DataIC50: 162nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Exscientia

US Patent
LigandPNGBDBM626036(US11786528, Example 15)
Affinity DataIC50: 253nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Exscientia

US Patent
LigandPNGBDBM626148(US11786528, Example 35)
Affinity DataIC50: 290nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
Exscientia

US Patent
LigandPNGBDBM626022(US11786528, Example 11)
Affinity DataIC50: 350nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Exscientia

US Patent
LigandPNGBDBM626148(US11786528, Example 35)
Affinity DataIC50: 530nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2023
Entry Details
US Patent

Displayed 1 to 50 (of 79 total ) | Next | Last >>
Jump to: