Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 12794
TargetProlyl hydroxylase EGLN2(Human)
Fibrogen

US Patent
LigandPNGBDBM240987(US9409892, 82 | US20250099455, Compound Formula I)
Affinity DataIC50: 700nMAssay Description:Enzyme activity is determined by capturing 14CO2 using an assay described by Kivirikko and Myllyla (1982, Methods Enzymol. 82:245-304). Assay reactio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetProlyl hydroxylase EGLN2(Human)
Fibrogen

US Patent
LigandPNGBDBM240987(US9409892, 82 | US20250099455, Compound Formula I)
Affinity DataIC50: 910nMAssay Description:Enzyme activity is determined by capturing 14CO2 using an assay described by Kivirikko and Myllyla (1982, Methods Enzymol. 82:245-304). Assay reactio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEgl nine homolog 1(Human)
Fibrogen

US Patent
LigandPNGBDBM240987(US9409892, 82 | US20250099455, Compound Formula I)
Affinity DataIC50: 1.69E+4nMAssay Description:Enzyme activity is determined by capturing 14CO2 using an assay described by Kivirikko and Myllyla (1982, Methods Enzymol. 82:245-304). Assay reactio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent

TargetEgl nine homolog 1(Human)
Fibrogen

US Patent
LigandPNGBDBM240987(US9409892, 82 | US20250099455, Compound Formula I)
Affinity DataIC50: 2.04E+4nMAssay Description:Enzyme activity is determined by capturing 14CO2 using an assay described by Kivirikko and Myllyla (1982, Methods Enzymol. 82:245-304). Assay reactio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2025
Entry Details
US Patent