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Report error Found 177 Enz. Inhib. hit(s) with all data for entry = 13562
LigandChemical structure of BindingDB Monomer ID 803969BDBM803969(US20260124222, Compound I-177)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803970BDBM803970(US20260124222, Compound I-178)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803967BDBM803967(US20260124222, Compound I-175)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803965BDBM803965(US20260124222, Compound I-173)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803966BDBM803966(US20260124222, Compound I-174)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803963BDBM803963(US20260124222, Compound I-171)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803964BDBM803964(US20260124222, Compound I-172)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803961BDBM803961(US20260124222, Compound I-169)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803962BDBM803962(US20260124222, Compound I-170)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803957BDBM803957(US20260124222, Compound I-165)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803958BDBM803958(US20260124222, Compound I-166)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803955BDBM803955(US20260124222, Compound I-163)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803956BDBM803956(US20260124222, Compound I-164)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803986BDBM803986(US20260124222, Compound I-194)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803983BDBM803983(US20260124222, Compound I-191)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803984BDBM803984(US20260124222, Compound I-192)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803981BDBM803981(US20260124222, Compound I-189)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803982BDBM803982(US20260124222, Compound I-190)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803979BDBM803979(US20260124222, Compound I-187)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803980BDBM803980(US20260124222, Compound I-188)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803978BDBM803978(US20260124222, Compound I-186)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803975BDBM803975(US20260124222, Compound I-183)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803976BDBM803976(US20260124222, Compound I-184)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803974BDBM803974(US20260124222, Compound I-182)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803972BDBM803972(US20260124222, Compound I-180)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 804002BDBM804002(US20260124222, Compound I-210)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803999BDBM803999(US20260124222, Compound I-207)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803998BDBM803998(US20260124222, Compound I-206)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803991BDBM803991(US20260124222, Compound I-199)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803992BDBM803992(US20260124222, Compound I-200)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803989BDBM803989(US20260124222, Compound I-197)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803990BDBM803990(US20260124222, Compound I-198)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK3 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803987BDBM803987(US20260124222, Compound I-195)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803988BDBM803988(US20260124222, Compound I-196)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 804003BDBM804003(US20260124222, Compound I-211)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit Tyk2 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 804004BDBM804004(US20260124222, Compound I-212)
Affinity DataIC50: 400nMAssay Description:Compounds of Formula I were screened for their ability to inhibit JAK1 using the general enzyme inhibition assay method, in which the assay mixture c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803856BDBM803856(US20260124222, Compound I-29)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803855BDBM803855(US20260124222, Compound I-28)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803858BDBM803858(US20260124222, Compound I-31)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803857BDBM803857(US20260124222, Compound I-30)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803852BDBM803852(US20260124222, Compound I-25)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803851BDBM803851(US20260124222, Compound I-24)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803854BDBM803854(US20260124222, Compound I-27)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803853BDBM803853(US20260124222, Compound I-26)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803848BDBM803848(US20260124222, Compound I-21)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803847BDBM803847(US20260124222, Compound I-20)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803850BDBM803850(US20260124222, Compound I-23)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803849BDBM803849(US20260124222, Compound I-22)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803867BDBM803867(US20260124222, Compound I-40)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 803869BDBM803869(US20260124222, Compound I-42)
Affinity DataIC50: 400nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/16/2026
Entry Details
US Patent

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